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Penicillamine increases free copper and enhances oxidative stress in the brain of toxic milk mice PMID 22629446
Octanoic acid
HIF signaling overactivation inhibits lateral line neuromast development through Wnt in zebrafish PMID 38097093
Structural and functional basis for (S)
SMO Protein
Halo tag TMR (solution)
AG
Mechanism of the thermogenic effect of Metabolite 2 (BTS 54 505), a major pharmacologically active metabolite of the novel anti
Novel Thio
4,4'
Bioactive terpenoids from the fruits of Aphanamixis grandifolia PMID 23772699
Asic1
GPRC5D as a novel target for the treatment of multiple myeloma a narrative review PMID 38307865
Amidinomycin from Streptomyces kasugaensis producing kasugamycin PMID 4975521
Mechanism
BCR
POC1 中心粒蛋白 B（POC1B）基因
Efficacy of Leukadherin
Doxofylline
HA/Hemagglutinin 蛋白, H1N1 (ACF54598, HEK293, His)
Activation of an AKT/FOXM1/STMN1 pathway drives resistance to tyrosine kinase inhibitors in lung cancer PMID 28850563
Cephalomannine 71610
Contribution of Cage
MCE
Long
FOLR1 Human Pre
Synthesis and structure
Anti
Decumbenine 76733
Anti
Increased intestinal permeability and downregulation of absorptive ion transporters Nhe3, Dra, and Sglt1 contribute to diarrhea during Clostridioides difficile infection PMID 37350393
Multifunctional neuroprotective effect of Withanone, a compound from Withania somnifera roots in alleviating cognitive dysfunction PMID 29108796
3,4
Cyclophilin A
Rohinitib 1139253
Discovery of Novel Coumarin
MCE
Myricanol represses renal fibrosis by activating TFAM and ZNRF1 to inhibit tubular epithelial cells ferroptosis PMID 39349116
The effects of photodynamic therapy on leukemia cells mediated by KillerRed, a genetically encoded fluorescent protein photosensitizer PMID 31590660
Calcrl
G 蛋白偶联受体 68（GPR68）基因
Antibacterial agent 96
Eicosatrienoic acid enhances the quality of in vitro matured porcine oocytes by reducing PRKN
P1788
Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic
Extended steroid profiling in H295R cells provides deeper insight into chemical
Biotin
HVEM/TNFRSF14 蛋白, Human (Biotinylated, HEK293, Fc
Gamma
MALT1 inhibitor MI
Complexins cytosolic proteins that regulate SNAP receptor function PMID 7553862
GSK572A
S100 钙结合蛋白 A12（S100A12）基因
PLLA3000
Oxaprozin
SM
Gna14
Anti
GNF
2,8
Epha2
Differential effects of two protein tyrosine kinase inhibitors, tyrphostin and genistein, on human bone cell proliferation as compared with differentiation PMID 9701629
Identification of Phosphorylation Consensus Sequences and Endogenous Neuronal Substrates of the Psychiatric Risk Kinase TNIK PMID 26645429
N
Oleyl Mesylate
Bromo
Amifloxacin (Win49375，氨氟沙星)
1
Carboxymethyl
Long term usage of dexamethasone accelerating accelerates the initiation of osteoarthritis via enhancing chondrocyte apoptosis and the extracellular matrix calcification and apoptosis of chondrocytes PMID 34803488
Negamycin induces translational stalling and miscoding by binding to the small subunit head domain of the Escherichia coli ribosome PMID 25368144
CRBN ligand
The protein level and transcription activity of activating transcription factor 1 is regulated by prolyl isomerase Pin1 in nasopharyngeal carcinoma progression PMID 28032861
Disruption of the SIRT1/PI3K/AKT Signaling Axis Mediates Fluoride
Synthesis and preliminary evaluation of 3
Ror1
TGF beta 1 抗体 (YA6435)（TGF beta 1 Antibody (YA6435)）
Bidirectional modulation of glycolysis using a multifunctional nanocomposite hydrogel promotes bone fracture healing in type 2 diabetes mellitus PMID 40256330
XY25026
(R)
Design and Synthesis of Novel and Selective Glycine Transporter
m
LMPTP inhibitor 1 1908414
The fully synthetic glycopeptide MAG
Fosl2
MCE
PD
N,N
BMP4 Signaling Acts via dual
Melatonin alleviates chronic stress
MACF1
Discovery of a Low Toxicity O
GRB2 is a BECN1 interacting protein that regulates autophagy PMID 38182563
SST1 receptor antagonist
Ethanol induces necroptosis in gastric epithelial cells in vitro PMID 33686694
MCE
9
含三方基序 60（TRIM60）基因
Label
MCE
Design, synthesis, and biological evaluation of 3
CRBN ligand
Discovery and Characterization of Potent, Efficacious, Orally Available Antimalarial Plasmepsin X Inhibitors and Preclinical Safety Assessment of UCB7362 PMID 36216349
In Vitro Delivery of mTOR inhibitors by Kidney
MCE
磷酸甘油酸脱氢酶（PHGDH）基因
Metabotropic glutamatergic receptors and their ligands in drug addiction PMID 24362085
TNFSF18
DRAM1 plays a tumor suppressor role in clear cell renal cell carcinoma through modulating Akt signaling PMID 35299128
Prkx Rat Pre
Sodium α
Potent cytotoxic rocaglamide derivatives from the fruits of Amoora cucullata PMID 16946551
HSF1 Pathway Inhibitor Clinical Candidate (CCT361814/NXP800) Developed from a Phenotypic Screen as a Potential Treatment for Refractory Ovarian Cancer and Other Malignancies PMID 37017629
MCE
Design and development of 5'
SHK1112218
Targeting the CXCR7 pathway with TC14012 to inhibit endothelial necroptosis and lung cancer metastasis PMID 40049294
Nucleos(t)ide analogs for hepatitis B virus infection differentially regulate the growth factor signaling in hepatocytes PMID 38180972
7
Tandospirone hydrochloride 99095
Viloxazine in the Management of CNS Disorders A Historical Overview and Current Status PMID 34003459
Salvianolic acid B protects against myocardial ischaemia
Ipsoprubart 3035552
F12 抗体 (YA7927)（F12 Antibody (YA7927)）
hsa
iASPP is essential for HIF
Inhibitory Effects of Isobavachalcone on Tau Protein Aggregation, Tau Phosphorylation, and Oligomeric Tau
Stable Cyclometalated Gold(III) Complex Engaging Isoquinoline Derivative and Disulfur Ligand Elicits Necroptosis
ZINC09875266
Transcription factor Zhx2 is a checkpoint that programs macrophage polarization and antitumor response PMID 37582865
Efficacy and Safety Exposure
抗病毒类药库
Thyroid stimulating hormone aggravates diabetic retinopathy through the mitochondrial apoptotic pathway PMID 34435365
Discovery of tetrandrine derivatives as tumor migration, invasion and angiogenesis inhibitors PMID 32599368
Bone morphogenetic protein
Rapirosiran sodium 2755197
Sbf1
基质金属肽酶 1（Mmp1）基因
Inhibition of gut
Bis
TCS 2314 317353
BO3482 198013
The antinociceptive effect of 1
SRP
5’
SPK
Cga
EP12 2882916
Tetramethylammonium hexafluorophosphate 558
Lipokine 5
白细胞介素 12B（IL12B）基因
GNE684 2438637
Ccne2 Rat Pre
Phosphatidylinositol 3
Effect of guaifenesin on cough reflex sensitivity PMID 14665498
TBAJ
KPI10
Discovery of novel sophocarpine derivatives as potential dual Bcl
C3C 抗体 (YA3594)（C3C Antibody (YA3594)）
LMPTP
Augmentation of the gastric mucosal defense mechanism induced by KW
Rilapladib 412950
LMPTP
Membrane Remodeling and Stimulation of Aggregation Following α
CD103
Amino
MLR
AR
Thrombomodulin 蛋白, Human (HEK293, His)
Pharmacokinetic evaluation of thiacetazone PMID 8888068
HA/Hemagglutinin 蛋白, H1N1 (AFR75881, HEK293, His)
Effects of Livagen peptide on chromatin activation in lymphocytes from old people PMID 12533768
Fmoc
H
GIT1
Xanthine oxidase
Spasmolytic effects of nonprenylated rotenoid constituents of Boerhaavia diffusa roots PMID 16792408
Card10 is a novel caspase recruitment domain/membrane
FOSL2 Human Pre
Cinnamomum zeylanicum extract 84649
A novel therapeutic target in various lung diseases airway proteases and protease
Highlights of the DNA cutters a short history of the restriction enzymes PMID 24141096
Discovery of novel pyridazinone derivatives as EGFRWT/ EGFRT790M kinase inhibitors; design, synthesis, antitumor evaluation, and molecular dynamic simulations PMID 41520616
Visualization of phagosomal hydrogen peroxide production by a novel fluorescent probe that is localized via SNAP
H
KPI 10
Boc
Fmoc
Discovery and characterization of Z1 an imipridone
Immunogenicity of the ALLAVGATK (gp100[17
2'
PSB
In vitro activities of iboga alkaloid congeners coronaridine and 18
MRLB
Clec7a Rat Pre
SESN2 prevents the slow
Pharmacological properties of tracazolate a new non
onion root tips
CF
Serrumab
Antitubercular constituents from the stem wood of Cinnamomum kotoense PMID 16180806
Polyacrylate
Klc1 Mouse Pre
WK500B 2253985
Syringetin 4423
Isopropyl myristate
Dexmedetomidine alleviated sepsis‑induced myocardial ferroptosis and septic heart injury PMID 32377745
Cyclophilin D plays a critical role in the survival of senescent cells PMID 39448884
Z
Deoxyadenosine diphosphate sodium 402491
benzaldehyde
An orally available small molecule BCL6 inhibitor effectively suppresses diffuse large B cell lymphoma cells growth in vitro and in vivo PMID 34990752
Apoc3
Sanggenol P (桑根酮醇P)
BAYV
Kat6a
Gly
Synthesis, Computational Insights, and Evaluation of Novel Sigma Receptors Ligands PMID 37155827
Phospho
Effects of MCI
中心体蛋白 72（CEP72）基因
LRP4 Human Pre
A Dendritic Cell
Delphinidin 3
Androgen receptor
Silver Nanoparticle
Hexyl salicylate
Silencing of the lncRNA TUG1 attenuates the epithelial
Modulation of FLT3
Construction of 3
Current methods to analyze lysosome morphology, positioning, motility and function PMID 35343629
Influenza virus
Conduritol B tetraacetate 25348
Cannabisin D from Sinomenium Acutum Inhibits Proliferation and Migration of Glioblastoma Cells through MAPKs Signaling PMID 33076708
The localization of messenger ribonucleic acids for somatostatin receptors 1, 2, and 3 in rat testis PMID 9421433
Design and structure
Ganglioside GT1b suppresses immunoglobulin production by human peripheral blood mononuclear cells PMID 10233751
Effect of 17beta
Pituitary and hypothalamic somatostatin receptor subtype messenger ribonucleic acid expression in the food
RP5171
A novel peptide TCL6148 induces ferroptosis via the GOT1/GPX4 pathway to enhance sunitinib sensitivity in renal cell carcinoma PMID 40379184
Activity of the phenothiazine methdilazine alone or in combination with isoniazid or streptomycin against Mycobacterium tuberculosis in mice PMID 19696152
Phytanic acid methyl ester 1118
H
Chenodeoxycholyl
Musashi 1/Msi1 抗体 (YA5255)（Musashi 1/Msi1 Antibody (YA5255)）
DMAC
Boc
34th Annual Meeting & Pre
Identification of multiple somatostatin receptors in the rat somatosensory cortex during development PMID 10805921
Development of a potent and selective GPR7 (NPBW1) agonist a systematic structure
Boc
Differential expression of multiple somatostatin receptors in the rat cerebellum during development PMID 9166718
Comparison of cell
CRBN ligand
Apotracker Red 2889374
Anti
赖氨酸甲基转移酶 2A（KMT2A）基因
N
STXBP2 Human Pre
CEP164 抗体 (YA8913)（CEP164 Antibody (YA8913)）
MK
NBzF
Lemairamin 29946
EZM0414 2411748
Adamantyl
NaBr
Downregulation of MCT4 for lactate exchange promotes the cytotoxicity of NK cells in breast carcinoma PMID 30051648
ClpP agonist 1 2761081
N
MCE
Sec18/NSF
Terbucarb
Crp
2
MAP3K14
LSD1/KDM1A
Anti
SCH 430765 405057
MRLB223
HSR
Neocaesalpin L 952473
Ibrutinib Inhibits BMX
Amithiozone
Methylcobalamin hydrate 288315
RO 5073012 1020814
Proadifen
Pyristriatins A and B Pyridino
hsa
Inhibiting the IGF
MK0536
Ac
MDL12330A 40297
(1E,4E)
radionuclide
Cbz
HRH3 抗体 (YA2701)（HRH3 Antibody (YA2701)）
Maytansinoid
Homogentisic acid
TEM8 marks neovasculogenic tumor
Human pyruvate kinase M2 a multifunctional protein PMID 20857498
NAD+ Metabolism Maintains the Homeostasis of Decidual Macrophages in Early Pregnancy PMID 40471104
P2X7 receptor promotes migration and invasion of non
Comparable In Vitro Activities of Second
A recombinant human immunoglobulin with coherent avidity to hepatitis B virus surface antigens of various viral genotypes and clinical mutants PMID 32790777
Ald
Ppib Rat Pre
Asb13 Rat Pre
Rad21 Mouse Pre
Paeoniae Radix Rubra extract attenuates cerebral ischemia injury by inhibiting ferroptosis and activating autophagy through the PI3K/Akt signalling pathway PMID 37172921
Pharmacological activation of TGR5 promotes intestinal growth via a GLP
Lucidadiol 252351
5
Phosphatidylglycerols (egg) sodium salt 383907
ABRO1 promotes NLRP3 inflammasome activation through regulation of NLRP3 deubiquitination PMID 30787184
Fibroblast Growth Factor Receptor 4 Promotes Triple
poly ADP ribose polymerase
A wearable device for continuous immunoassay
A fully enzymatic method for site
Oncogenic and prognostic role of CKAP2L in hepatocellular carcinoma PMID 32509063
Protective effects of growth hormone
Synthesis of 2
5,6,7,4'
Z
MGMT
Scarf1
H
KP 544 393856
FXR as a pivotal role linking JNK and G0s2 mitigates triptolide
Fmoc
RBC
PERK controls bone homeostasis through the regulation of osteoclast differentiation and function PMID 33051453
Benzofuran
Antiparasitic agent
CRAMP analog having potent antibiotic activity without hemolytic activity PMID 12144503
Cefepime 88040
Pharmacological inhibition of BMK1 suppresses tumor growth through promyelocytic leukemia protein PMID 20832753
Down
Recombinant human erythropoietin protects the myocardium from ischemia
DL
MCE
Propargyl
Structure
Htr1b Rat Pre
RPA70 抗体 (YA5280)（RPA70 Antibody (YA5280)）
WU
Design and synthesis of ROCK2
Inhibition of cytochrome P450 by proadifen diminishes the excitability of brain serotonin neurons in rats PMID 30431437
DCLK
Sodium 2
Structure
Novel 18beta
EGFR signaling confers resistance to BET inhibition in hepatocellular carcinoma through stabilizing oncogenic MYC PMID 30770740
84294
in advanced prostate cancer
Mmrn1 Rat Pre
Monoamine Oxidase
The Alzheimer's disease drug candidate J147 decreases blood plasma fatty acid levels via modulation of AMPK/ACC1 signaling in the liver PMID 35051863
Cytochrome P450 inhibitor
MCE
Fursultiamine 804
One Year of Abaloparatide, a Selective Activator of the PTH1 Receptor, Increased Bone Formation and Bone Mass in Osteopenic Ovariectomized Rats Without Increasing Bone Resorption PMID 27748532
Levonorgestrel
MCE
2
canavan disease
Antimalarial agent 16 2773408
Discovery of new quinazoline derivatives as irreversible dual EGFR/HER2 inhibitors and their anticancer activities
Translocation of HIV TAT peptide and analogues induced by multiplexed membrane and cytoskeletal interactions PMID 21969533
In vivo and in vitro cardiovascular effects of Papuan taipan (Oxyuranus scutellatus) venom Exploring sudden collapse PMID 22771951
Chicoric Acid Attenuated Renal Tubular Injury in HFD
H
AGL 2043 226717
核糖核苷酸还原酶催化亚基 M1（RRM1）基因
Neogenin interacts with hemojuvelin through its two membrane
lung function
A thalamic
磷脂酶 A2 X 组（PLA2G10）基因
siRNA delivery into tumor cells by cationic cholesterol derivative
Galactosyl cholesterol
Luxdegalutamide 2750830
Mapping the active site of angiotensin
SARS
Umbelliferone
Raltegravir is a potent inhibitor of XMRV, a virus implicated in prostate cancer and chronic fatigue syndrome PMID 20376347
Calamenene 483
ND
WL 12
Proteasome inhibitor MG132 induces apoptosis in human osteosarcoma U2OS cells PMID 34002651
Oxodipine 90729
DS 28120313
GDC
3
growth factor
Metoclopramide dihydrochloride 2576
DL
HG
1,3
Trastuzumab
DL
Synthesis and in vitro study of pseudo
Deferasirox
A novel retinoid, 4
binding peptide
LRRFIP2 Human Pre
ARV 766
Cyclopalladated primary amines a preliminary study of antiproliferative activity through apoptosis induction PMID 25063943
Osteoporosis
Unveiling the role of RAC3 in the growth and invasion of cisplatin
Further exploring the tolerant region II Identification of 2,4,5
VTCN1
From docking false
CRBN ligand
RO27
CD20
HSDB 7455
5,6
Urotensin I, a CRF
Succinyl hydroxamates as potent and selective non
GPR40 Activator 3 2980
Comparative Pharmacology of a Bis
Trigalacturonic acid 6037
MCE
BMS986365
Dual Pro
Znrf3 Mouse Pre
Nor
DN 1679
antiacid
Palonosetron
Lipopolysaccharide downregulates the expression of p53 through activation of MDM2 and enhances activation of nuclear factor
Discovery of chebulagic acid and punicalagin as novel allosteric inhibitors of SARS
SiR
ATP
DS
mmu
A novel androgen receptor antagonist JJ
BMS
GDP366 501698
viral DNA
(2E)
Ghrelin administered spinally increases the blood glucose level in mice PMID 24472858
Parsaclisib Is a Next
BAY 771
An in vitro study on interaction of anisodine and monocrotaline with organic cation transporters of the SLC22 and SLC47 families PMID 31514980
5
Tetrachyrin 73483
BRD4
The agonist activities of the putative antipsychotic agents, L
Bronchodilator and anti
Androsin alleviates non
FAK inhibitor 5 1426683
HEMTAC WEE1 degrader
Isobavachalcone suppresses expression of inducible nitric oxide synthase induced by Toll
BACE
Cyclic GMP phosphodiesterase inhibitors. 2. Requirement of 6
Flavokawin C 56798
Chemical genetics reveals a kinase
Wortmannin binds specifically to 1
12(S)
Milestones to the Discovery of T
Pharmacological characterization of recombinant human and rat P2X receptor subtypes PMID 10440098
PGHS
68Ga
Caficrestat 1355612
Ferrostatin
Discovery of (S)
Besifloxacin Hydrochloride 405165
Systemic blockade of P2X7 receptor protects against sepsis
Efanesoctocog alfa the renaissance of Factor VIII replacement therapy PMID 38356459
Aloxistatin 88321
A super
destructase
PKM zeta maintains late long
Discovery of seven
Adverse events that are associated with the selective estrogen receptor modulator levormeloxifene in an aborted phase III osteoporosis treatment study PMID 12237621
TNP
14
AS602801 Sensitizes Ovarian Cancer Stem Cells to Paclitaxel by Down
NMB Human Pre
High
Methylboronic acid pinacol ester
Simultaneous characterisation of multiple Mahonia fortunei bioactive compounds in rat plasma by UPLC
anticoagulative
MCE
Thalidomide
Phosphodiesterase inhibitory activity of the flavonoids and xanthones from Anaxagorea luzonensis PMID 25920267
Besifloxacin, a novel fluoroquinolone antimicrobial agent, exhibits potent inhibition of pro
H
The dual peroxisome proliferator
lesions
Mivavotinib monohydrochloride 1952251
Octanorcucurbitane and cucurbitane triterpenoids from the tubers of Hemsleya endecaphylla with HIV
Collagen cross
Dextran sulfate modulates MAP kinase signaling and reduces endothelial injury in a rat aortic clamping model PMID 19563964
血管内皮锌指 1（VEZF1）基因
(Rac)
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