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Inhibitory effect of antineoplaston A
Ac
Map1lc3b
LCK 原癌基因，Src 家族酪氨酸激酶（LCK）基因
Discovery of potent and stable conformationally constrained analogues of the MCH R1 antagonist SB
Boc
Effects of dopamine D1 receptor agonists in rats trained to discriminate dihydrexidine PMID 16575553
Bcl2 样2（Bcl2l2）基因
Prap1
Co
F2 R 样凝血酶或胰蛋白酶受体 3（F2rl3）基因
Old Friends With New Faces Are Sodium Channel Blockers the Future of Adjunct Pain Medication Management? PMID 28842369
Gpr3
In Vitro Activity of Bedaquiline against Nontuberculous Mycobacteria in China PMID 28242674
Genkwanin inhibits proinflammatory mediators mainly through the regulation of miR
Arrest of preterm labor in rat and mouse by an oral and selective nonprostanoid antagonist of the prostaglandin F2alpha receptor (FP) PMID 17618756
D
Amn
Psmd14
Fibroblast growth factor 10 attenuates chronic obstructive pulmonary disease by protecting against glycocalyx impairment and endothelial apoptosis PMID 36183124
Methyl tridecanoate 1731
Comparison of the cytotoxicity in vitro of temozolomide and dacarbazine, prodrugs of 3
Activin RIB/ALK
阿特拉斯蛋白 GTPase 1（ATL1）基因
Meeting report 31st International Conference on Antiviral Research PMID 30086336
Elinzanetant (NT
cross
Effects of endogenous agonists, glycine and D
Myristic acid reduces skin inflammation and nociception PMID 34811755
Fulvotomentoside B 1021184
EETs Reduction Contributes to Granulosa Cell Senescence and Endometriosis
Neotame (GMP Like)
LAH4 enhances CD8+ T cell immunity of protein/peptide
Wls
ISIS 329993 827355
A Novel Agonist of the Type 1 Lysophosphatidic Acid Receptor (LPA1), UCM
NCX
Phaseoloideside C (榼藤子皂苷C)
Polysimiaric acid B
Polysimiaric acid A
Planchol E
NM102
IBPR002
Cappariloside A
DBCO
Phos
LCD36
cFLFLF
12
NOTA
UNC7242
Cofilin
Antiparasitic agent
Production of plasmid DNA for pharmaceutical use PMID 17875478
Nsmaf
Endothelium
Exonuclease
Potent and selective cyclohexyl
Gonadotropin
4
In vitro antibacterial activity and beta
ALK
Preclinical candidate for the treatment of visceral leishmaniasis that acts through proteasome inhibition PMID 30962368
Gastrointestinal absorption of sulfaguanidine in neonatal and adult rats PMID 3820055
Forkhead box M1 inhibits endothelial cell apoptosis and cell
MCE
The σ 1 receptor agonist 4
Differential roles of 3
Association of cyclic adenosine monophosphate with permeability barrier homeostasis of murine skin PMID 14962102
The Regulation of Cerebral Lymphatic Drainage in the Transverse Sinus Region of the Mouse Brain PMID 39289863
Morusin suppresses breast cancer cell growth in vitro and in vivo through C/EBPβ and PPARγ mediated lipoapoptosis PMID 26538209
The 5
Discovery of ATR kinase inhibitor berzosertib (VX
Distinct features of bivalent direct thrombin inhibitors, hirudin and bivalirudin, revealed by clot waveform analysis and enzyme kinetics in coagulation assays PMID 31366633
Recombinant soluble gp130 protein reduces DEN
A novel and sensitive UPLC
Defensins natural component of human innate immunity PMID 23756165
3,4
Zatonacaftor 2301945
Trans
Comparison of calcipotriol with selected metabolites and analogues of vitamin D3 effects on cell growth regulation in vitro and calcium metabolism in vivo PMID 8396769
RNA 聚合酶 II 相关蛋白 2（RPAP2）基因
APOH
Heterologous expression of a novel galactose
MKC
Intragastric and intraoesophageal pH monitoring in duodenal ulcerpatients effect of the new histamine H2
FLT3 inhibitors induce p53 instability, driven by STAT5/MDM2/p53 competitive interactions in acute myeloid leukemia PMID 39756787
IKZF2
RPS6KB2
A novel tubulin inhibitor, No.07, shows anti
Antagonists of the platelet P2T receptor a novel approach to antithrombotic therapy PMID 9925726
Discovery and Characterization of Fluorine
Kinsenoside Suppresses DGAT1
2,3
CRBN ligand
PI3K
Wilforic acid A 193684
Novel mammalian cell cycle inhibitors, tryprostatins A, B and other diketopiperazines produced by Aspergillus fumigatus. II. Physico
Mixed Lineage Kinase
Discovery and Characterization of Novel BLIMP
Sulfaethidole 94
Uncovering the rewired IAP
Sufu limits sepsis
Epilepsy in adults PMID 30686584
Multiscale imaging of colitis in mice using confocal laser endomicroscopy, light
Characterization of a novel cyclin
Tyrosinase
Inhibition of ICAM1 diminishes stemness and enhances antitumor immunity in glioblastoma via β
Discovery of INCB159020, an Orally Bioavailable KRAS G12D Inhibitor PMID 39772605
Adenosine Uptake through the Nucleoside Transporter ENT1 Suppresses Antitumor Immunity and T
Opioid Receptor
Rab5a
2
Discovery of heterocyclic nonacetamide synaptic vesicle protein 2A (SV2A) ligands with single
Impacts of Intralipid on Nanodrug Abraxane Therapy and on the Innate Immune System PMID 32071352
Neuregulin
Bis
New Insights into the Virulence Traits and Antibiotic Resistance of Enterococci Isolated from Diverse Probiotic Products PMID 33807433
MCE
p53 (17
[Experimental osteoarthritis and its course when treated with S
Repurposing Nitazoxanide for Potential Treatment of Rare Disease Lymphangioleiomyomatosis PMID 39456169
P
Tesidolumab (LFG316) for treatment of C5
BGTC
LYN
Dipeptide PA3264 derived from rare and endangered Squama Manis is a novel bioactive peptide for the treatment of triple
Ecabapide, a novel gastroprokinetic agent, ameliorates gastric emptying of stroke
Brominated Azaphilones from the Sponge
HIF
MP
Lymph node fibroblastic reticular cells preserve a tolerogenic niche in allograft transplantation through laminin α4 PMID 35775481
Sialidase
Lacto
MCE
Co
A sensitive WST
Benzene
High
MAO
Il2ra
Hexadecatetraenoic acid
RGS2 is an innate immune checkpoint for suppressing Gαq
A20 inhibits periodontal bone resorption and NLRP3
LPL Receptor
Compositional analyses of a human menopausal gonadotrophin preparation extracted from urine (menotropin). Identification of some of its major impurities PMID 14680547
Encainide
Pinaverium impurity 1
Levonadifloxacin arginine hydrate ((S)
Light
Phosphodiesterase 5 inhibitor mirodenafil ameliorates Alzheimer
(S,S)
Phenylpropiophenone derivatives as potential anticancer agents synthesis, biological evaluation and quantitative structure
Aspulvinones Suppress Postprandial Hyperglycemia as Potent α
Fluorphine 6440
CBGA
Protocol for modeling acquired resistance to targeted therapeutics in adherent and suspension cancer cell lines via in situ resistance assay PMID 39369385
Benzylamine hydrochloride 3287
TACA
The analgesic effect of carbiphene hydrochloride PMID 4921303
RTA
The pharmacology of tacrine at N
Epsiprantel 98123
5
5
Corydalis Saxicola Bunting Total Alkaloid Eliminates Porphyromonas gingivalis strain 33277 Internalized into Macrophages by Inhibition of TLR2 PMID 37914020
Methocarbamol
RAS
Nonsteroidal antiinflammatory drug hydroxamic acids. Dual inhibitors of both cyclooxygenase and 5
Pentagalloylglucose suppresses the growth and migration of human nasopharyngeal cancer cells via the GSK3β/β
Spectral characteristics of voltage
MLS000545091 322666
Ptpn5 Mouse Pre
A rapid method of concentrating proteins in small volumes with high recovery using Sephadex G
Tinazoline 62882
OX40
Furfuryl
Discovery of a potential anti
Anoikis Resistance as a Further Trait of Acidic
κOR
TTPAL promotes gastric tumorigenesis by directly targeting NNMT to activate PI3K/AKT signaling PMID 34642500
Naringenin as a phytogenic adjuvant systematically enhances the protective efficacy of H9N2 inactivated vaccine through coordinated innate
3,3'
Potential synergic mechanism of Wutou
Reversal of activity
Bioactive chemical constituents from the root bark of Morus australis PMID 27908762
Polyprenol (13~21) (Polyprenol mixture (13~21))
Dedicator of Cytokinesis 5 Regulates Keratinocyte Function and Promotes Diabetic Wound Healing PMID 33627322
Pennogenin 3
The discovery of PLK4 inhibitors (E)
Anastrozole impurity 1 (Standard)
Toward the Selective Inhibition of G Proteins Total Synthesis of a Simplified YM
[Effect of dimephosphon on the inflammatory reaction] PMID 3410029
Jingzhaotoxin
Asialoglycoprotein receptor 1 functions as a tumor suppressor in liver cancer via inhibition of STAT3 PMID 36043912
Doxapram hydrochloride hydrate 7081
Folate
Haloxyfop
Royal jelly acid, 10
Calcitriol in cancer treatment from the lab to the clinic PMID 15026558
DHTP is an allosteric inhibitor of the kinesin
MCE
The natural product trienomycin A is a STAT3 pathway inhibitor that exhibits potent in vitro and in vivo efficacy against pancreatic cancer PMID 33687738
MCE
ITK inhibition induced in vitro and in vivo anti
Expression of the FOS proto
SMYD2 aggravates gastrointestinal stromal tumor via upregulation of EZH2 and downregulation of TET1 PMID 35668081
AZD8931, an equipotent, reversible inhibitor of signaling by epidermal growth factor receptor, ERBB2 (HER2), and ERBB3 a unique agent for simultaneous ERBB receptor blockade in cancer PMID 20145185
5
Mechanism of smooth muscle relaxation by tiropramide PMID 6114146
[Effect of hypoxia on the expression of macrophage migration inhibitory factor (MIF) in rat vascular smooth muscle cells] PMID 19462902
Analytical method development and preformulation stability studies of L
(2S,3R)
Increase in the levels of chaperone proteins by exposure to beta
hsa
Octahydroaminoacridine succinate
Antibacterial agent 265
钙结合蛋白 4（CABP4）基因
5
Mutagenic evaluation of the hair
The bacterial serine protease inhibitor ecotin inhibits neutrophil elastase enzymatic activity in cystic fibrosis sputa PMID 39444402
P53/PANK1/miR
Functionally active cyclin
Luteoloside pretreatment attenuates anoxia
NB4
Tripotassium phosphate 7778
dTAG
Amn
(S)
Mki67
MCE
Tomentosin Reduces Behavior Deficits and Neuroinflammatory Response in MPTP
Doxorubicin
A Placebo
Metabolic Enzyme SLC27A5 Regulates PIP4K2A pre
Oral treatment with a novel small molecule alpha 4 integrin antagonist, AJM300, prevents the development of experimental colitis in mice PMID 23623333
Identification of novel LRRK2 inhibitors by structure
Comparison of antimicrobial activities and resistance mechanisms of eravacycline and tigecycline against clinical Acinetobacter baumannii isolates in China PMID 39380684
Target of rapamycin coordinates auxin are involved in exogenous melatonin regulated low temperature tolerance in cucumber seedlings PMID 39182426
Epigenetic reactivation of tumor suppressor genes by a novel small
Development and evaluation of topical formulations for a novel skin whitening agent (AP736) using Hansen solubility parameters and PEG
Defining the mechanism of action and enzymatic selectivity of psammaplin A against its epigenetic targets PMID 22280363
Discovery of phenylalanine derivatives as potent HIV
Zamifenacin (UK
Interaction potential of Carmegliptin with P
Others 抑制剂
CD4 antigen
Adrenocorticotropin(1
Discovery of a bifunctional PKMYT1
Thiamethoxam
mutant repeat expansion transcripts
Steroidal saponins from Asparagus curillus fruits PMID 17405104
The pharmacokinetics of penamecillin PMID 19108231
PTP1B
IL
Epicoprostanol found in adipocere from five human autopsies PMID 9397400
XCL1 and XCR1 in the immune system PMID 22100876
Activity of fusidic acid against extracellular and intracellular Staphylococcus aureus influence of pH and comparison with linezolid and clindamycin PMID 21546626
Discovery and optimization of boronic acid based inhibitors of autotaxin PMID 20536182
Kynuramine, a fluorescent substrate and probe of plasma amine oxidase PMID 562342
Antitumor agent
Mitophagy
Enhancing Aqueous Solubility and Antibacterial Activity of Curcumin by Complexing with Cell
5
Lck
Treatment for ovarian hyperstimulation syndrome using an oral dopamine prodrug, docarpamine PMID 14503971
Inhibition of NF
Gardenoside ameliorates inflammation and inhibits ECM degradation in IL
Analogs of methyl
Calpastatin subdomain B 128578
DL
Bis
Activity of cephalosporin CXA
Development of visible
Alterations in the molecular regulation of mitochondrial metabolism in human alveolar epithelial cells in response to cigarette
dASK1
Heavy ion radiation
Synthesis and structure
Bladder cancer detection using a peptide substrate of the 20S proteasome PMID 27326540
Silybin
CDK4/6 inhibitor palbociclib suppresses IgE
CRBN ligand
Identification of binding sites on the regulatory A subunit of protein phosphatase 2A for the catalytic C subunit and for tumor antigens of simian virus 40 and polyomavirus PMID 1328865
CBP/p300
GABAergic Interneuron and Neurotransmission Are mTOR
Her4.3+ radial glial cells maintain the brain vascular network through activation of Wnt signaling PMID 39019216
Cyclohexanoyl coenzyme A 5960
Novel hybrid molecules based on 15
A novel dual NLRP1 and NLRP3 inflammasome inhibitor for the treatment of inflammatory diseases PMID 37360982
Molecular basis of the structure and function of H1 hemagglutinin of influenza virus PMID 22728439
NDR1/FBXO11 promotes phosphorylation
Effects of the 5
Synthesis and SAR study of 4
MS437 541535
Virtual screening
Psiguadials A and B, two novel meroterpenoids with unusual skeletons from the leaves of Psidium guajava PMID 20929258
IGF1R/ARRB1 Mediated Regulation of ERK and cAMP Pathways in Response to Aβ Unfolds Novel Therapeutic Avenue in Alzheimer's Disease PMID 39969678
多形性胶质母细胞瘤
Identification and synthesis of quinolizidines with anti
YOD1 sustains NOD2
Protection against monocrotaline
MS67
The SARS
all
Alpha
Carbonic anhydrase IX
Hepatoprotective effect of pinostrobin against thioacetamide
Sanfetrinem 156769
MYC 原癌基因，bHLH 转录因子（MYC）基因
Inhibition of LPS
PF
EGFR
PC3 sections
Cdc7
Intracellular degradation of two structurally different polyhydroxyalkanoic acids accumulated in Pseudomonas putida and Pseudomonas citronellolis from mixtures of octanoic acid and 5
PL
EGFR
CTTHWGFTLC, CYCLIC 244082
5
11(S)
肽酶抑制因子 16（PI16）基因
Structure
Isocarlinoside
XW
degrader
Discovery of a Small
N
Hydantion indolinones as AANAT inhibitors PMID 41176235
Design, synthesis and evaluation of novel HIV
CRBN ligand
18 1 (8
Targeted Protein Degradation by Chimeric Compounds using Hydrophobic E3 Ligands and Adamantane Moiety PMID 32106507
Synthesis, biological evaluation and molecular docking studies of pyrazole derivatives coupling with a thiourea moiety as novel CDKs inhibitors PMID 23933045
Synthesis and Biological Evaluation of Heterocycle
MAO
CRBN ligand
Budipine 57982
2
Growth inhibition of mouse autochthonous skin cancer by oral administration of new serine protease inhibitor ONO
Discovery of M Protease Inhibitors Encoded by SARS
STAG1 vulnerabilities for exploiting cohesin synthetic lethality in STAG2
CFL1 Human Pre
Sigma
MCE
MCE
Macrophage secretory IL
FR900359 107530
Design of fast
Enhanced fluorescence lifetime imaging microscopy denoising via principal component analysis PMID 40060483
Amitivir 111393
AHR/cyp1b1 signaling
Concurrent inhibition of CDK2 adds to the anti
Crystal structure of human aldehyde dehydrogenase 1A3 complexed with NAD+ and retinoic acid PMID 27759097
3’
1,2
BRD4
Small
TLR7/8 agonists activate a mild immune response in rabbits through TLR8 but not TLR7 PMID 25131730
Optically active selenium
Combining adoptive NK cell infusion with a dopamine
6
A smart tablet
MCE
Partial inhibition of adipose CIDEC improves insulin sensitivity and increases energy expenditure in high
RAF1 蛋白, Human (Y340D, Y341D, sf9, His, GST)
ARN
Effect of cyclodextrins on the complexation and transdermal delivery of bupranolol through rat skin PMID 15129982
NMI promotes cell proliferation through TGFβ/Smad pathway by upregulating STAT1 in colorectal cancer PMID 31230364
Regiocontrol of Soybean Lipoxygenase Oxygenation. Application to the Chemoenzymatic Synthesis of Methyl 15(S)
MCE
Ca2+ channel antagonist U
Epitalon 307297
Decursin inhibits vasculogenesis in early tumor progression by suppression of endothelial progenitor cell differentiation and function PMID 22298358
TNF
Purification, bioactivity and application of maltobionic acid in active films PMID 38188310
Therapeutic potential of IKK
Potent, Selective, and Cell Active Protein Arginine Methyltransferase 5 (PRMT5) Inhibitor Developed by Structure
Exosomal Prolactin
The Bengamides A Mini
N
N
Family
[Effect of a water
Bis
Z
Bekanamycin 4696
F 盒蛋白 4（FBXO4）基因
Design, Synthesis, and Biological Activity of Novel Thiazole Sulfonamide Derivatives as Potent Fungicide Candidates against Sclerotinia sclerotiorum PMID 41187972
Org
CD38 分子（CD38）基因
Alliin 556
In vivo determination of the volatile metabolites of saprotroph fungi by comprehensive two
Earlier onset of chemotherapy
Differences between in
4,8
From Bench to Clinic A Nitroreductase Rv3368c
Thiazole
Efficient antibacterial agents a review of the synthesis, biological evaluation and mechanism of pleuromutilin derivatives PMID 24200363
Molecular dynamics simulation of a DOPA/ST monolayer on the Au(111) surface PMID 23936904
TATA 盒结合蛋白相关因子 1 样（TAF1L）基因
Therapeutic effects of the allosteric protein tyrosine phosphatase 1B inhibitor KY
[BMIM]Cl (1
Indolinyl
Glisoprenins C, D and E, new inhibitors of appressorium formation in Magnaporthe grisea, from cultures of Gliocladium roseum. 1. Production and biological activities PMID 9544931
SUCNR1 regulates insulin secretion and glucose elevates the succinate response in people with prediabetes PMID 38713514
c
A strategy for constructing large protein interaction maps using the yeast two
ca2
Rfc1
A Pdx
MCE
Glycofurol 31692
Lysine methyltransferase SMYD2 promotes cyst growth in autosomal dominant polycystic kidney disease PMID 28604386
MCE
Rodorubicin 96497
Adipose invariant NKT cells interact with CD1d
Mouse models of hepatocellular carcinoma an overview and highlights for immunotherapy research PMID 29904153
MCL0020 475498
Lgr6
Tap1
MCE
Development of mercapto
MCE
Identification of benzodiazepine Ro5
Transmembrane AMPA receptor regulatory proteins and cornichon
VC1052
Synthesis and antiprotozoal activity of cationic 1,4
CRBN ligand
Synthesis, biological evaluation, and molecular docking studies of N
Stigmalactam from Orophea enterocarpa induces human cancer cell apoptosis via a mitochondrial pathway PMID 25556482
Soluble epoxide hydrolase inhibitor 1241826
Ibetazol, a novel inhibitor of importin β1
RA signaling pathway combined with Wnt signaling pathway regulates human
AMPA receptor potentiators application for depression and Parkinson's disease PMID 17504104
Binding of diarrheic shellfish poisoning toxins to okadaic acid binding proteins purified from the sponge Halichondria okadai PMID 20863709
Ovalbumin
Deuteration Strategy
Cathepsin S therapeutic, diagnostic, and prognostic potential PMID 25872877
Identification of inhibitors targeting the FLT3
Lead suppresses perlecan expression via EGFR
Identification of a novel boronic acid as a potent, selective, and orally active hormone sensitive lipase inhibitor PMID 27338659
Hit
Azithromycin modulates Teff/Treg balance in retinal inflammation via the mTOR signaling pathway PMID 34600916
MC70 potentiates doxorubicin efficacy in colon and breast cancer in vitro treatment PMID 21925160
Pdx1
TDIQ hydrochloride 15052
Immunotoxicity of Benzothiazole on Mytilus Edulis Following In Vitro Exposure of Hemocytes PMID 30701043
Nitroxynil 1689
Antidiarrheal activity of α
ACT 128800
Dehydroepiandrosterone sulfate 651
MCE
Genome
CISD3 is a prognostic biomarker and therapeutic target in pan
Isocryptotanshinone Induced Apoptosis and Activated MAPK Signaling in Human Breast Cancer MCF
EED
Emtricitabine, a new antiretroviral agent with activity against HIV and hepatitis B virus PMID 16323102
Inhibition of DNA methylation reverses norepinephrine
PSI
Antiinflammatory constituents of Celastrus orbiculatus inhibit the NF
Human fucosyltransferase IX specificity towards N
Pyrazole
WEE1 Kinase Inhibitor AZD1775 Has Preclinical Efficacy in LKB1
Herbal compound cepharanthine attenuates inflammatory arthritis by blocking macrophage M1 polarization PMID 37976601
SPRYD4 Human Pre
Avibactam sodium hydrate 2938989
CRBN ligand
Ptpn5
(S)
Involvement of TLR4 signaling regulated
Quantification of α
Effect of Fidaxomicin versus Vancomycin on Susceptibility to Intestinal Colonization with Vancomycin
New natural urease inhibitors from Ranunculus repens PMID 16570500
In Vitro Activity of Sulopenem, an Oral Penem, against Urinary Isolates of Escherichia coli PMID 30397056
Diethylphosphine oxide 7215
Conventional and atypical antipsychotics in the elderly a review PMID 17535043
Targeting erbB Pathways in Breast Cancer Dual Kinase Inhibition for Brain Metastasis and Prevention of p185HER2/Neu Tumor Development PMID 39493351
Antibacterial Activity of Linezolid against Gram
Development of natural products for anti
酸性磷酸酶 6，溶血磷脂（ACP6）基因
克立昔单抗
AFN 941
YAP knockdown in combination with ferroptosis induction increases the sensitivity of HOS human osteosarcoma cells to pyropheophorbide
Redefining the major peanut allergens PMID 22948807
Wee1
Biotinylated quercetin as an intrinsic photoaffinity proteomics probe for the identification of quercetin target proteins PMID 21798748
Hepoxilin A3 formation in the rat pineal gland selectively utilizes (12S)
Inhibition of protein synthesis by spectinomycin PMID 5318092
雌激素受体 1（ESR1）基因
The exploration of aza
A reappraisal of the mucoactive activity and clinical efficacy of bromhexine PMID 28331610
SOX10 deficiency
Pharmacokinetics and Pharmacodynamics of Azeloprazole Sodium, a Novel Proton Pump Inhibitor, in Healthy Japanese Volunteers PMID 29193126
REDV 107978
5
Local anaesthetic pain relief therapy In vitro and in vivo evaluation of a nanotechnological formulation co
Gamitrinib TPP 1131626
The pan
Preventing protein adsorption and macrophage uptake of gold nanoparticles via a hydrophobic shield PMID 23009596
2
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