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UBP710 1333111
Filastatin 431996
Development of a sphingosine kinase 1 specific small
Synthesis of novel 2,4
Pyridinone derivatives specific human immunodeficiency virus type 1 reverse transcriptase inhibitors with antiviral activity PMID 1713693
Anti
EP
Cardiovascular events and safety outcomes associated with remdesivir using a World Health Organization international pharmacovigilance database PMID 34719115
Gitoformate 10176
PD
Synthesis and antitumor activity of some new xanthotoxin derivatives PMID 19217697
New biologically active compounds from Kenyan propolis PMID 20079813
Tubulin polymerization
Genotoxicity of 1,3
4
Combinatorial allosteric modulation of agonist response in a self
Pharmacokinetics and pharmacodynamics of HTD1801 (berberine ursodeoxycholate, BUDCA) in patients with hyperlipidemia PMID 33183320
p38 MAPK
Targeting PIK3CG in Combination with Paclitaxel as a Potential Therapeutic Regimen in Claudin
GLP
Structure
The antitumor effect of lowered doses of cytostatics combined with new analogs of vitamin D in mice PMID 17970085
Eriocalyxin B, a novel autophagy inducer, exerts anti
Chitohexaose activates macrophages by alternate pathway through TLR4 and blocks endotoxemia PMID 22654663
A glutamine metabolic switch supports erythropoiesis PMID 39541460
The plant alkaloid voacamine induces apoptosis
Discovery of a first
Hydrouracil
Fluorescence Anisotropy Studies on Bodipy (Pyrromethene 546) Dye as a Novel Thermal Probe PMID 35059931
AF
Luminacin C1 251449
A comparative study of triacylglycerol composition in Chinese human milk within different lactation stages and imported infant formula by SFC coupled with Q
Ethoxyquin dimer 74681
Capacitative and 1
L
Estrogen inhibits autophagy and promotes growth of endometrial cancer by promoting glutamine metabolism PMID 31429768
Estradiol
Suramin sodium salt 129
Regulation of cancer cell death by a novel compound, C604, in a c
Distearoylphosphatidylserine
Acetylvardenafil 1261351
Triiodothyronine and dexamethasone alter potassium channel expression and promote electrophysiological maturation of human
Identification of a Highly Cooperative PROTAC Degrader Targeting GTP
Structure
SR 717
Characterisation of a new chimeric ligand for galanin receptors galanin(1
Regulation of exocrine pancreatic secretion by cerebral TRH and CGRP role of VIP, muscarinic, and adrenergic pathways PMID 8447406
Tissue kallikrein mK13 is a candidate processing enzyme for the precursor of interleukin
MCE
Boc
Synthesis and formulation studies of griseofulvin analogues with improved solubility and metabolic stability PMID 28258034
DNA damage and cell cycle arrest induced by 2
Update on the development of antagonists of chemoattractant receptor
Tolterodine is a novel candidate for assessing CYP3A4 activity through metabolic volatiles to predict drug responses PMID 39828876
Virtual and In Vitro Antiviral Screening Revive Therapeutic Drugs for COVID
Targeting Class I Histone Deacetylases Triggers Antitumor Responses in Colorectal Cancer In Vitro and In Vivo PMID 41486684
Activation of the Aryl Hydrocarbon Receptor by 10
DHMB 4055
Wall shear stress modulates metabolic pathways in endothelial cells PMID 39832080
ST1926, a novel and orally active retinoid
Development of an ICOSL and BAFF bispecific inhibitor AMG 570 for systemic lupus erythematosus treatment PMID 30789152
Mal
Pradimicin Q, a new pradimicin aglycone, with alpha
Pharmacokinetics of N
Study on Biological Characteristics and Mechanism of Paclitaxel Induced Drug Resistance in Endometrial Carcinoma Cells PMID 30175145
Tuftsin diacetate 72103
MTSSL 81213
Anti
Fatty Acid Transport Proteins Targeting FATP2 as a Gatekeeper Involved in the Transport of Exogenous Fatty Acids PMID 27446528
MCE
Leptin and insulin synergize with PIK3CA mutation to enhance PD
The therapeutic effects of tuberostemonine against cigarette smoke
Diethylhomospermine 119422
16 0 Caproylamine PE
Directed differentiation of human
OMDM
Fluvastatin sodium 93957
远西方印迹法
Dalotuzumab 1005389
Metabolism distribution and excretion of a matrix metalloproteinase
Phenolphthalein glucuronide sodium 6820
Epigenetic regulation of beta
hsa
AMPK activator C2 1428422
Biotin
Enhanced kinase translocation reporters for simultaneous real
In vivo pharmacodynamics of ceftobiprole against multiple bacterial pathogens in murine thigh and lung infection models PMID 18676887
光滑的，卷曲的类受体（Smo）基因
D
MCE
Research progress of LSD1
Brahma links the SWI/SNF chromatin
MCE
Benzimidazoisoquinolines a new class of rapidly metabolized aryl hydrocarbon receptor (AhR) ligands that induce AhR
Opromazine hydrochloride 316
AH 8529 41805
SDZ 216
Photoaffinity label for the alpha 1
(1R,2S,7R)
CP
hsa
Cyclophilin D is required for mitochondrial removal by autophagy in cardiac cells PMID 20364102
Boc
Novel non
Flumizole 36740
DHODH
Discovery of amino
A novel histone deacetylase inhibitor, CG200745, potentiates anticancer effect of docetaxel in prostate cancer via decreasing Mcl
3,6
Identification of Gαi3 as a promising molecular oncotarget of pancreatic cancer PMID 39349432
Dehydrotrametenolic acid 6879
3
Fluorescence
Tanshinone IIA alleviates pulmonary fibrosis by modulating glutamine metabolic reprogramming based on [U
MAT2A
Single cell RNA
Analog of somatostatin vapreotide exhibits biological effects in vitro via interaction with neurokinin
HER2 breast cancer
MCE
Structure
Optical control of butyrylcholinesterase (BChE) activity via photoswitchable azobenzene for potential treatment of Alzheimer's disease PMID 39348751
Sialidase inhibitors attenuate pulmonary fibrosis in a mouse model PMID 29118338
Br
Triterpene glycosides of Siraitia grosvenori inhibit rat intestinal maltase and suppress the rise in blood glucose level after a single oral administration of maltose in rats PMID 15826043
δ Opioid Receptor Agonism Preserves the Retinal Pigmented Epithelial Cell Tight Junctions and Ameliorates the Retinopathy in Experimental Diabetes PMID 31529081
Dihydromaniwamycin E 3033567
A Novel CD206 Targeting Peptide Inhibits Bleomycin
Bioactive lignans from Peperomia heyneana PMID 17291043
Binding domains of the oxytocin receptor for the selective oxytocin receptor antagonist barusiban in comparison to the agonists oxytocin and carbetocin PMID 15740719
MCE
Components of the DNA methylation system of chromatin control are RNA
RET
ME3277, a GPIIb/IIIa antagonist reduces cerebral infarction without enhancing intracranial hemorrhage in photothrombotic occlusion of rabbit middle cerebral artery PMID 10894182
Guanfacine 29110
Hepatotoxicity of Two Progoitrin
The fungal natural product azaphilone
Isolation and purification of a modified phenazine, griseoluteic acid, produced by Streptomyces griseoluteus P510 PMID 21262358
19(S),20(R)
Assessing Supersaturation and Its Impact on In Vivo Bioavailability of a Low
Dipeptidase‑2 is a prognostic marker in lung adenocarcinoma that is correlated with its sensitivity to cisplatin PMID 37449493
Carcinogenicity study of doxefazepam administered in the diet to Sprague
5A2
Intranasal administration of the TLR2 agonist Pam2Cys provides rapid protection against influenza in mice PMID 22823162
Biochemical characterization of tirabrutinib and other irreversible inhibitors of Bruton's tyrosine kinase reveals differences in on
Rhodamine 800 as a probe of energization of cells and tissues in the near
MALT1
Carborane
MCE
Dynamic regulation of N6,2'
16 0 PE
Stimulation of choleragen enzymatic activities by GTP and two soluble proteins purified from bovine brain PMID 3123477
Ro
Lodenafil 139755
Inostamycin, an inhibitor of cytidine 5'
Synthesis and in vitro antiproliferative activity of C5
Characterization and DNA
Drug susceptibility and the potential for drug
CITFA 2379989
The Novel Glutamine Antagonist Prodrug JHU395 Has Antitumor Activity in Malignant Peripheral Nerve Sheath Tumor PMID 31594823
Molybdic acid, 85% MoO3 basis 7782
Sinapine thiocyanate 7431
Dose
Antiviral activity of lambda
DBCO
13
18 1 MPB PE 384835
Mycobacterium tuberculosis CrgA Forms a Dimeric Structure with Its Transmembrane Domain Sandwiched between Cytoplasmic and Periplasmic β
Sarracenin 59653
Viloxazine Increases Extracellular Concentrations of Norepinephrine, Dopamine, and Serotonin in the Rat Prefrontal Cortex at Doses Relevant for the Treatment of Attention
Piperazine A Promising Scaffold with Analgesic and Anti
Small molecule
[Ala92]
Discovery of 2
GDC
MCE
Acetyl angiotensinogen (1
Development of a novel N14
Antioxidant, anti
Crozbaciclib fumarate 2567494
Btk Inhibitors A Medicinal Chemistry and Drug Delivery Perspective PMID 34299259
L
Machine
Design and synthesis of caffeoyl
AChE
Synthesis of Quinoline
mmu
Optimization of 2
α
Terallethrin 15589
Microcystin
Val
MTOB sodium 51828
Discovery of Novel Resorcinol Dibenzyl Ethers Targeting the Programmed Cell Death
2
Nefazodone a new antidepressant PMID 8748566
del(8p) and TNFRSF10B loss are associated with a poor prognosis and resistance to fludarabine in chronic lymphocytic leukemia PMID 37752286
Development of small molecule inhibitors targeting RNA helicase DHX33 as anti
Upregulation of PREX1 Expression by POU2F2 Promotes the Malignant Progression of Acute Myeloid Leukemia via the mTOR Pathway PMID 40317800
SLAMF3 promotes Th17 differentiation and is reversed by iguratimod through JAK1/STAT3 pathway in primary Sjögren's syndrome PMID 38061117
Naratriptan biological profile in animal models relevant to migraine PMID 9170336
Quinazolinone Compounds Have Potent Antiviral Activity against Zika and Dengue Virus PMID 37506506
AChE
NSC 245214 31554
Chromostatin (bovine) 133633
Tc
The G132S Mutation Enhances the Resistance of Mycobacterium tuberculosis β
Tyrosinase
Effects of Complex I Inhibition on the Architecture of Neural Rosettes Differentiated from Human
Inhibition of TRPM8 by the urinary tract analgesic drug phenazopyridine PMID 36657655
Effects of threo
阿维巴坦钠二水合物
Assay of protein and peptide adducts of cholesterol ozonolysis products by hydrophobic and click enrichment methods PMID 25185119
MCE
Efficacy of Acetylshikonin in Preventing Obesity and Hepatic Steatosis in db/db Mice PMID 27483220
Pentaethylene glycol (Standard)
MCE
Gut microbiota modulation through Akkermansia spp. supplementation increases CAR
NTRK fusion promotes tumor migration and invasion through epithelial
Post
Piperlongumine (piplartine) and analogues Antiproliferative microtubule
SKP
S 38093, a histamine H3 antagonist/inverse agonist, promotes hippocampal neurogenesis and improves context discrimination task in aged mice PMID 28218311
SFTPA1 Human Pre
MCE
Bidirectional modulation of HIF
Activation of mitophagy by rapamycin eliminated the accumulation of TDP
Reverse
m6A Methylation of Precursor
父系表达 10（PEG10）基因
Toxicological evaluations of the benzodiazepine doxefazepam PMID 2568837
4
Novel truncating variants in CTNNB1 cause familial exudative vitreoretinopathy PMID 35361685
Rosuvastatin protects against coronary microembolization
HAP1 PARP16 KO cells
Lactose (Standard)
BCM
Blood schizontocidal and gametocytocidal activity of 3
2
1,2
Preparative liquid chromatography PMID 12236522
Discovery of Novel Dihydrothiopyrano[4,3
8
Electron tunneling from electronically excited states of isolated bisdisulizole
MCE
AZD1080, a novel GSK3 inhibitor, rescues synaptic plasticity deficits in rodent brain and exhibits peripheral target engagement in humans PMID 23410232
MCE
Poly
Metabolomic analysis of murine tissues infected with Brucella melitensis PMID 39869554
Novel Cinnamic Acid Derivatives Containing Naproxen as NLRP3 Inhibitors Synthesis and Evaluation of Their Biological Activity PMID 39737737
IL
N
TNFRSF17
Angiotensin
CSTF2
N
Characterization of a new aryl
ARMCX3 regulates ROS signaling, affects neural differentiation and inflammatory microenvironment in dental pulp stem cells PMID 39296219
Sulfanitran
Safety, Tolerability, and Pharmacokinetics of Ibuprofenamine Hydrochloride Spray (NSAIDs), a New Drug for Rheumatoid Arthritis and Osteoarthritis, in Healthy Chinese Subjects PMID 33628011
Imaging protein synthesis in cells and tissues with an alkyne analog of puromycin PMID 22160674
Hypotensive effect and toxicology of total alkaloids and veratramine from roots and rhizomes of Veratrum nigrum L. in spontaneously hypertensive rats PMID 18771011
Studies on the relation of chemical structure to glycogenolytic activity in the brain PMID 4637949
pH
Resveratrol inhibits paclitaxel
CaMK1b/PNCK
Gastric antisecretory effects of esaprazole in rats PMID 1356865
Doxorubicin
Hepatitis B Virus Core Protein Mediates the Upregulation of C5α Receptor 1 via NF
IHMT
MCE
Identification of a Novel Protein Phosphatase 2A Activator, PPA24, as a Potential Therapeutic for FOLFOX
Cyclin N
N
Food intake in baboons effects of a long
radioimmunotherapy
Binding site and inhibitory mechanism of the mambalgin
Receptor binding profile of neuropeptide gamma and its fragments comparison with the nonmammalian peptides carassin and ranakinin at three mammalian tachykinin receptors PMID 8234024
Live imaging of osteoclast inhibition by bisphosphonates in a medaka osteoporosis model PMID 26704995
Adam12
DMT
SPTSSA Human Pre
Butylamine
Nfrkb Rat Pre
Angiotensin II type 2 receptor pharmacological agonist, C21, reduces the inflammation and pain hypersensitivity in mice with joint inflammatory pain PMID 35724606
MCE
Circular RNA circCLASP2 promotes nasopharyngeal carcinoma progression through binding to DHX9 to enhance PCMT1 translation PMID 40050914
Interplay between gut microbial communities and metabolites modulates pan
FITC
1,2,3,4,6,7,8
LncRNA MIAT suppresses inflammation in LPS
Emricasan Ameliorates Portal Hypertension and Liver Fibrosis in Cirrhotic Rats Through a Hepatocyte
The effect of a xanthine derivative, 1
Effect of butobendin on dopamine beta
The Biochemical and Clinical Perspectives of Lactate Dehydrogenase An Enzyme of Active Metabolism PMID 31886754
SNF9007 a novel analgesic that acts simultaneously at delta 1, delta 2 and mu opioid receptors PMID 8182541
Identification of an Antiviral Compound from the Pandemic Response Box that Efficiently Inhibits SARS
An agonistic monoclonal antibody against DR5 induces ROS production, sustained JNK activation and Endo G release in Jurkat leukemia cells PMID 19468286
MSA 2
Synthesis of 2,3,6,7
Functional targeting of the TGF
Amlodipine, an anti
LysRs
Ravoxertinib hydrochloride 2070009
hsa
5
Tyrosine ethyl ester 34081
MCE
HuR
Pharmacological modulation of gp130 signalling enhances Achilles tendon repair by regulating tenocyte migration and collagen synthesis via SHP2
LncRNA DIO3OS regulated by TGF
Methyl heptadecanoate
beclin 1（Becn1）基因
Spatial organization of lysosomal exocytosis relies on membrane tension gradients PMID 36800388
Effects of bromopride on abdominal wall healing with induced peritoneal sepsis after segmental colectomy and colonic anastomosis in rats PMID 22042104
Microbiome Metabolite
AKR7A3 Human Pre
Hsp90 beta 抗体 (YA6336)（Hsp90 beta Antibody (YA6336)）
Discovery of a Hidden Pocket beneath the NES Groove by Novel Noncovalent CRM1 Inhibitors PMID 38105606
m
Small molecule discoidin domain receptor kinase inhibitors and potential medical applications PMID 25569119
Leptomycin B is an inhibitor of nuclear export inhibition of nucleo
Discovery, Structure
Nogo
RG7204 (PLX4032), a selective BRAFV600E inhibitor, displays potent antitumor activity in preclinical melanoma models PMID 20551065
MCE
Time
An alternative Alcian Blue dye variant for the evaluation of fetal cartilage PMID 17410541
JNJ 26481585
LTBP1 plays a potential bridge between depressive disorder and glioblastoma PMID 33059753
Transmembrane modification of tumor vascular targeting peptide A7R as molecular cargo delivery tool PMID 38412651
Intratumoral delivery of a highly active form of XCL1 enhances antitumor CTL responses through recruitment of CXCL9
Danger
Bimolane in vitro inhibitor of human topoisomerase II PMID 9461029
MCE
DL
Disulfiram treatment suppresses antibody
Paroxetine alleviates T lymphocyte activation and infiltration to joints of collagen
MDC/CCL22 蛋白, Rat
MAP4K
PIK3CA mutations contribute to fulvestrant resistance in ER
Influenza A variants with reduced susceptibility to baloxavir isolated from Japanese patients are fit and transmit through respiratory droplets PMID 31768027
ICAM
Anti
Guanosine
CREBBP
Selective inhibition of BET bromodomains PMID 20871596
The therapeutic value of XL388 in human glioma cells PMID 33159013
MCE
Luoshi Neiyi Prescription inhibits estradiol synthesis and inflammation in endometriosis through the HIF1A/EZH2/SF
Solid
SCARF1 Human Pre
Alpha5 nicotine acetylcholine receptor subunit promotes intrahepatic cholangiocarcinoma metastasis PMID 38453934
Pin4
Antiviral evaluation of hydroxyethylamine analogs Inhibitors of SARS
Vigilin interacts with ER
N,N
2'
Investigating the Anticancer Activity of Isatin/Dihydropyrazole Hybrids PMID 30996798
Inhibition of translation in eukaryotic systems by harringtonine PMID 319998
BCMA
Deferasirox shows in vitro and in vivo antileukemic effects on murine leukemic cell lines regardless of iron status PMID 23415674
IL
长穗桑提取物 (Morus wittiorum Hand.
Optimisation of LRRK2 inhibitors and assessment of functional efficacy in cell
Targeting YAP1
Role of topical peptides in preventing or treating aged skin PMID 19570099
Design, synthesis and antimycobacterial activity of less lipophilic Q203 derivatives containing alkaline fused ring moieties PMID 30692025
The ALK inhibitor PF
SARM regulates CCL5 production in macrophages by promoting the recruitment of transcription factors and RNA polymerase II to the Ccl5 promoter PMID 24711619
Photosensitive and dual
N,N
First Penicillin
Diethylstilbestrol and risk of psychiatric disorders a critical review and new insights PMID 21428730
IL
Neurokinin receptor antagonists as potential non
MCE
Cardioprotection by a nonerythropoietic, tissue
Maprotiline Suppresses Cholesterol Biosynthesis and Hepatocellular Carcinoma Progression Through Direct Targeting of CRABP1 PMID 34093212
Ebelactone, an inhibitor of esterase, produced by actinomycetes PMID 7251497
Mechanism of action and in vivo role of platelet
alpha
Levobetaxolol 93221
Pharmacokinetics of oral pridinol Results of a randomized, crossover bioequivalence trial in healthy subjects PMID 33835016
Near
Quantitation of serum pregnanediol
MRS1845 544478
PRB3 Human Pre
Exosomal circ
Neuregulin
Perindoprilat
The mechanosensitive Piezo1 channel exacerbates myocardial ischaemia/reperfusion injury by activating caspase
Pleiotropic Effects of Influenza H1, H3, and B Baloxavir
Phenazone
MCE
Nicotinamide phosphoribosyl transferase
HIV
The Effects of an Albumin Binding Moiety on the Targeting and Pharmacokinetics of an Integrin αvβ6
Mono
COX
DNase I, Bovine pancreas
Avibactam sodium
BNP 抗体 (YA4345)（BNP Antibody (YA4345)）
Atypically Modified Carbapenem Antibiotics Display Improved Antimycobacterial Activity in the Absence of β
4
西那卡塞杂质杂质12
Measurement of Human Cytochrome P450 Enzyme Induction Based on Mesalazine and Mosapride Citrate Treatments Using a Luminescent Assay PMID 26336590
Nfrkb Mouse Pre
Proteotoxic stress
New
Phenazoviridin 155233
Aromadendrin 6
Nucleoporins shape germ granule architecture and balance small RNA silencing pathways PMID 39896640
Praeruptorin B 73069
hsa
Hsp90 beta 抗体 (YA5288)（Hsp90 beta Antibody (YA5288)）
MCE
hsa
β(3)
Dibenzosuberone 1210
Tetrahydrolipstatin
Binimetinib 606143
3',5'
1
18 0 EPC chloride 328268
Putrescine
TAT
PROTAC BTK Degrader
ELAVL4 蛋白, Human (His
FtsZ inhibitor
Micronutrient antioxidant supplementation alleviates valproic acid
(2
程序性细胞死亡 6（PDCD6）基因
Revaprazan hydrochloride 178307
甘油茶碱
Trandolaprilate 87679
(
SIRT6 Negatively Regulates Schwann Cells Dedifferentiation via Targeting c
Glycyrin 66056
Non
Stimulatory and inhibitory activity of STING ligands on tumor
硝苯醋磺胺
Inhibitory effects of antihistamines, diphenhydramine and chlorpheniramine, on proton currents in BV2 microglial cells PMID 28131782
MCE
MCE
NDRG1 Human Pre
POU 2 类同源框关联因子 1（POU2AF1）基因
Synthesis and biological evaluation of new steroidal pyridines as potential anti
Aminooxy
MCE
PTK6
THP
MCE
MCE
N2
内皮素1（Edn1）基因
Diosgenin attenuates non
L15 cells
Tyrosylprotein Sulfotransferase2
porphyrias
NXL
Tumor acidosis supports cancer cell lipid uptake via a rapid transporter
Dual modulation of cytotoxic and checkpoint receptors tunes the efficacy of adoptive Delta One T cell therapy against colorectal cancer PMID 40240620
RUVBL2
2
5
芬布芬 d<sub>9</sub>
Marsdenoside A 858360
HM30181 mesylate
十四烷基
OXA
WNT7B promotes cancer progression via WNT/β
Novel topoisomerase I inhibitors. Syntheses and biological evaluation of phosphorus substituted quinoline derivates with antiproliferative activity PMID 29501943
Dihydrozeatin riboside 22663
Obesity
c[Arg
PROTAC 20S proteasome subunit β5 degrader 1
英文化学名 (标准品)
MCE
CTLA
A tractable covalent linker strategy for the production of immunogenic antigen
N6
Disulfide
MCE
DSG4 Human Pre
NSC232003 1905453
4
Mannosamine–lipoic acid adduct
1,N6
Rlf
CSF2 promotes chemoresistance in colorectal cancer by regulating Notch pathway PMID 40202620
DSG4
JWZ
KT203 1402612
Hygromycin B (Standard)
Tert
IGF1 Receptor 抗体 (YA4905)（IGF1 Receptor Antibody (YA4905)）
DMBP 133156
Heclin 890605
S100 A8 抗体 (YA1170)（S100 A8 Antibody (YA1170)）
BMY
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