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ML095 (CID
Colchiceine 477
CPTP
RelB
MCE
N
biosensing
1,1'
Quercitrin 2''
Effects of transitory maternal pteroylglutamic acid (PGA) deficiency on respiratory control ratios, phosphorylative capacity, and cytochrome oxidase activities of mitochondria from rat embryos PMID 4336911
Argininic acid 157
DDPO
ProINDY
Triazolinone biphenylsulfonamides as angiotensin II receptor antagonists with high affinity for both the AT1 and AT2 subtypes PMID 7799397
4
Maleimide
Peimine 23496
1
Pck2 Rat Pre
A phase I clinical trial of novobiocin, a modulator of alkylating agent cytotoxicity PMID 1985770
Fatty Acid Synthase (FASN)
Stresscopin (human)
EIF1AX 蛋白, Human (His)
HOOC
Glycerol 3
MCE
MCE
Zilpaterol
Extracellular vesicles derived from CD4+ T cells carry DGKK to promote sepsis
Vonoprazan impurity 6
Discovery of ZX079 as a Dual PROTAC Degrader Targeting BRD4/CBP in Acute Myeloid Leukemia PMID 41701037
Fragment
Brazilin
Resistance to pyrimethamine/sulfadoxine in Plasmodium falciparum in 12 villages in north east Tanzania and a test of chlorproguanil/dapsone PMID 9088432
4
ML
Physical stabilisation of amorphous ketoconazole in solid dispersions with polyvinylpyrrolidone K25 PMID 11113645
PLXDC2 蛋白, Human (HEK293, His)
ZL 1218
Adafenoxate 82168
11(E),13(E)
大三叶升麻提取物 (Actaea heracleifolia (Kom.) J. Compton)
HHAT
Sulfo
Antibacterial agent 128
NPFF2
Rivaroxaban impurity 9
MAO
Design, Synthesis and Biological Evaluation of Novel and Potent Protein Arginine Methyltransferases 5 Inhibitors for Cancer Therapy PMID 36235174
MMB
Combating Autoimmune Diseases With Retinoic Acid Receptor
AD67
Drug intermediate
Targeted inhibition of YAP/TAZ alters the biological behaviours of keloid fibroblasts PMID 34623712
Idasanutlin (Standard)
3
Enhanced retention and anti
GC
p75NTR Promotes Astrocyte Proliferation in Response to Cortical Stab Wound PMID 33201418
Read
Pantoprazole impurity 26
Novel Nitrophenyl Substituted Anthranilic Diamide Derivatives Design, Synthesis, Selectivity, and Antiresistance PMID 37939255
Cell culture biology's new dimension PMID 12931155
肌细胞增强因子 2B（MEF2B）基因
PGF2α 1,15
Discovery of ganodecalone A, from Ganoderma calidophilum for the treatment of acute gastric ulcers by binding to ALOX5 via the MAPK/NF
Wallichoside 60657
Isotschimgin 62356
Micellar solubilization of timobesone acetate in aqueous and aqueous propylene glycol solutions of nonionic surfactants PMID 3247274
DL
Zebrafish models
GCN2
Tetrazolast 95104
Angeloyl
(R)
Antitrypanosomal agent 26
6
Bombesin receptor antagonist
iDeg
JC
8(R)
Anti
Dihydrotetrabenazine (DHTBZ)
E
SIBP
omega
Moroxydine hydrochloride 3160
千日红提取物 (Gomphrena globosa L.)
元宝草提取物 (Hypericum sampsonii Hance)
Amino
Regulated macrophage immune microenvironment in 3D printed scaffolds for bone tumor postoperative treatment PMID 35574049
Vbp1
Discovery of the novel antithrombotic agent 5
Synthesis and evaluation of indenopyrazoles as cyclin
Sec13
Tyrosinase
MCE
O2172
Tetramethylammonium iodide 75
Foeniculoside I
Ncf4 Mouse Pre
Rolzavosoritide 3067191
Lestaurtinib's antineoplastic activity converges on JAK/STAT signaling to inhibit treatment naïve and therapy resistant forms ovarian cancer PMID 40646138
Others 抑制剂
BRD9 ligand
AQX 1125
CD72 Human Pre
In vitro and in vivo activity of NY
Got2
1
MCE
Design, Synthesis, and Biological Evaluation of the First Inhibitors of Oncogenic CHD1L PMID 35192363
Inhibition of MAO A and B by some plant
(3S)
N
2’,3’,5’
CRBN ligand
Investigation of monotherapy and combined anticoronaviral therapies against feline coronavirus serotype II in vitro PMID 34676775
Prevascularized Hydrogel Enhancing Innervation and Repair of Full
Anti
Adenosine 5
MDC1
Apigenin 6
Preskimmianin (Preskimmianine，前茵芋碱)
Duloxetine impurity 1
MCE
Site
Omipalisib (Standard)
ZSCAN4 Human Pre
MCE
1,10
OC
MCE
Brevinin
Butropium bromide
CD73
CD73
cIAP
Antibacterial and antilarval compounds from marine gorgonian
S26131
Intratumor Mycoplasma promotes the initiation and progression of hepatocellular carcinoma PMID 38088929
Identification and characterization of triamcinolone acetonide, a microglial
Oridonin exerts anticonvulsant profile and neuroprotective activity in epileptic mice by inhibiting NLRP3
Feruloylputrescine 501
Inhibition of adenosine uptake in human erythrocytes by adenosine
Tiaprofenic acid
Prasugrel metabolite
4'
Osthole stimulates osteoblast differentiation and bone formation by activation of beta
And1 degrader 1
Efficient Generation of Small Intestinal Epithelial
喙荚鹰叶刺提取物 (Guilandina minax (Hance) G. P. Lewis)
tunicate
MCE
Selective inhibition of platelet n
Sensitivity to the two peptide bacteriocin plantaricin EF is dependent on CorC, a membrane
Apoa4
[Double blind controlled study of miroprofen in acute upper respiratory tract infections
醛脱氢酶 1 家族成员 A1（ALDH1A1）基因
Brca1 Rat Pre
Prevention of experimental acute otitis media with penicillin V PMID 2106761
3
The unique catalytic properties of PSAT1 mediate metabolic adaptation to glutamine blockade PMID 39192144
2′
Conjugated and unconjugated bilirubins in bile of humans and rhesus monkeys. Structure of adult human and rhesus
PfCLK3
New antibiotic, isohematinic acid. II. Physico
High
Propane
brain
百子莲提取物 (Agapanthus africanus Hoffmgg.)
(E/Z)
Protective functions of liver X receptor α on calcified aortic valve involvement of regulating endoplasmic reticulum
The selective sphingosine 1
Anxiolytic
Antitumor agent
Estradiol
Lemon Balm Extract
STING
2
OrangeIV 554
Pyridostigmine in the treatment of postural orthostatic tachycardia a single
Arbidol as a broad
2
Fatty acid transduction of nitric oxide signaling. Nitrolinoleic acid is a hydrophobically stabilized nitric oxide donor PMID 15764811
CD3G 抗体 (YA538)（CD3G Antibody (YA538)）
The Protective Effect of Hispidin against Hydrogen Peroxide
Doxorubicin
主题讲座
Tamapin, a venom peptide from the Indian red scorpion (Mesobuthus tamulus) that targets small conductance Ca2+
Fluvoxamine alleviates bleomycin
Bengamin hydrochloride (4
RET
2
DMBA
New structures and bioactivity properties of jasplakinolide (jaspamide) analogues from marine sponges PMID 20121114
Human PTH
Mianserin 24219
Discovery of Novel N
Ncoa6
KRASG12D
Dual anti
Antitumor effect of L
Bisdeoxycoelenterazine derivatives for improvement of bioluminescence resonance energy transfer assays PMID 17850082
The ZFHX3 (ATBF1) transcription factor induces PDGFRB, which activates ATM in the cytoplasm to protect cerebellar neurons from oxidative stress PMID 20876357
Pharmacological characterization of cinnamophilin, a novel dual inhibitor of thromboxane synthase and thromboxane A2 receptor PMID 8019768
Discovery and Development of 1
(20S) Ginsenoside Rh2 Inhibits STAT3/VEGF Signaling by Targeting Annexin A2 PMID 34502195
VCB
The protective effect of caffeic acid on global cerebral ischemia
Crotonamide (巴豆酰胺)
SCP
Terephthalaldehyde (Terephthalaldehyde)
Cadalene
CHF6001 I a novel highly potent and selective phosphodiesterase 4 inhibitor with robust anti
2
The effect of anti
5
Macrocyclic lathyrane type diterpene esters (jolkinols) from callus cultures and roots of Euphorbia lathyris PMID 6484031
Esculeoside A (番茄皂苷A)
Oligomeric self
Prdx6
MCE
2
Sin3a
Plasma concentrations and receptor binding of RU 486 and its metabolites in humans PMID 3560943
CHAF1A interacts with TCF4 to promote gastric carcinogenesis via upregulation of c
Idh3g
Nicotiflorin attenuates cell apoptosis in renal ischemia
USP26
Active ingredients Isorhamnetin of Croci Srigma inhibit stomach adenocarcinomas progression by MAPK/mTOR signaling pathway PMID 37537191
菟丝子提取物 (Cuscuta chinensis Lam.)
MCE
MED12 interacts with the heat
Lead Optimization Yields High Affinity Frizzled 7
RADX prevents genome instability by confining replication fork reversal to stalled forks PMID 34107305
Delayed Wound Healing in Heat Stable Antigen (HSA/CD24)
MCE
Hypotensive effects of [D
厚鳞柯提取物 (Lithocarpus pachylepis A. Camus)
MCE
MCE
酰基辅酶 A 脱氢酶短链/支链（ACADSB）基因
rel
HECT, UBA and WWE domain containing 1 represses cholesterol efflux during CD4+ T cell activation in Sjögren's syndrome PMID 37435494
DKK1, a negative regulator of Wnt signaling, is a target of the beta
Chaetomella acutiseta produces chaetomellic acids A and B which are reversible inhibitors of farnesyl
Plasma inhibitory activity (PIA) a pharmacodynamic assay reveals insights into the basis for cytotoxic response to FLT3 inhibitors PMID 16857987
Naringenin 4',7
Targeting internal ribosome entry site (IRES)
Synthesis and biological evaluation of 4
Msi1
PGE2 upregulates the Na+/K+ ATPase in HepG2 cells via EP4 receptors and intracellular calcium PMID 33444342
Vps41
Proadrenomedullin (1
SIK2 maintains breast cancer stemness by phosphorylating LRP6 and activating Wnt/β
Collapsin response mediator protein 2 (CRMP2) interacts with N
Ptgr2
A reptilian neurohypophysial hormone, mesotocin (Ile8
Design, synthesis and evaluation of semi
In vivo antitumoral activity of stem pineapple (Ananas comosus) bromelain PMID 17893836
Quinazoline derivatives as selective CYP1B1 inhibitors PMID 28259840
Identification of triazolopyridine derivatives as a new class of AhR agonists and evaluation of anti
Possible involvement of neuropeptide Y sub
Dibenzoylmethane Protects Against CCl4
Mearnsitrin
A new role for FGF2 as an endogenous inhibitor of anxiety PMID 19439615
Nizofenone, a neuroprotective drug, suppresses glutamate release and lactate accumulation PMID 7813567
1
Nsmaf
Disease
[Review [new antibiotics series III] micronomicin (author's transl)] PMID 7047790
New lanostanoids of Ganoderma tsugae PMID 10785428
Hbegf
Asgr2
Cyanoguanidine
MCE
Comparative antihypertensive effects of guanabenz and clonidine PMID 7037502
Aspartyl
Effects of crosstalk between steroid hormones mediated thyroid hormone in zebrafish exposed to 4
Fpr3
神经钙蛋白结合蛋白 1（CABIN1）基因
Tedisamil dihydrochloride 132523
Human H
dilation
CI572
Pseudomonas aeruginosa Induces Interferon
The SWI/SNF chromatin remodeling factor DPF3 regulates metastasis of ccRCC by modulating TGF
Trijugin
Antibacterial activity in vitro of sulbenicillin against mucoid and non
Burnettramic acid A
Chloroxylenol disrupts Rana chensinensis tadpoles metabolic homeostasis via gut microbiota
A Survey of Commercially Available Isomaltooligosaccharide
Transcriptional inhibition of cytochrome P4502E1 by a synthetic compound, YH439 PMID 8579361
The marine natural product manzamine A targets vacuolar ATPases and inhibits autophagy in pancreatic cancer cells PMID 24048269
Cletoquine
主题讲座
U2surp
含补丁域 1（PTCHD1）基因
Development of Simultaneous Drug Concentration Measurement Method Using an Automated Pretreatment Liquid Chromatography/Tandem Mass Spectrometry System for Therapeutic Drug Monitoring PMID 39339175
SL65.0155, a novel 5
Anti
Carvedilol impurity 1
The Role of Decoy Receptor DcR3 in Gastrointestinal Malignancy PMID 35813013
Mrap2
Clinical and laboratory studies of sodium diphenicillin. II. Clinical studies, with emphasis on the rate of disappearance of staphylococci from various lesions PMID 13999396
Spatial control of the TSC complex integrates insulin and nutrient regulation of mTORC1 at the lysosome PMID 24529379
Converting enzyme inhibitors and the role of the sulfhydryl group in the potentiation of exo
The antisecretory effects of zaltidine, a novel long
Fumagillol 108102
α
Methyl benzoate and cinnamate analogs as modulators of DNA methylation in hepatocellular carcinoma PMID 35451561
Nek2
PDCD4 Negatively Regulated Osteogenic Differentiation and Bone Defect Repair of Mesenchymal Stem Cells Through GSK
Gins2
Incorporation of synthetic 1,2
Discovery of WML
1,2,3
Eumenitin, a novel antimicrobial peptide from the venom of the solitary eumenine wasp Eumenes rubronotatus PMID 16762455
Visual Identification of Trichosporon asahii, a Gut Yeast Associated with Obesity, Using an Enzymatic NIR Fluorescent Probe PMID 35920602
Tissue distribution study of columbianadin and its active metabolite columbianetin in rats PMID 26115176
Development of C
Nr1i2
The Werner and Bloom syndrome proteins catalyze regression of a model replication fork PMID 17115688
JH
The pharmacological properties of seclazone (7
Nazartinib S
Thymosin β4 reverses phenotypic polarization of glial cells and cognitive impairment via negative regulation of NF
Identification and characterization of the ocular hypotensive efficacy of travoprost, a potent and selective FP prostaglandin receptor agonist, and AL
TAT
BRCA1 抗体 (YA819)（BRCA1 Antibody (YA819)）
Conserved patterns of transcriptional dysregulation, heterogeneity, and cell states in clear cell kidney cancer PMID 39792555
surface lipid
Benzo(a)pyrenediolepoxide
Alteminostat 1246374
N
Click
Degradation of parathion methyl in bovine milk by high
MFB
Targeting specific proteins for lysosomal proteolysis PMID 1801703
A Novel CSN5 Inhibitor Drives Tumor
NKP608 a selective NK
Normal development of mice and unimpaired cell adhesion/cell motility/actin
Discovery of novel osthole derivatives exerting anti
1
Safety evaluation study of lincomycin and spectinomycin hydrochloride intramuscular injection in chickens PMID 35169546
BGN
Improving flavor of summer Keemun black tea by solid
Chemistry and biochemistry of palm oil PMID 11106812
Maternal obesity interrupts the coordination of the unfolded protein response and heat shock response in the postnatal developing hypothalamus of male offspring in mice PMID 33636254
Hmgn2
Arl2
Inhibition of the replication of a hepatitis C virus
High
uPAR 蛋白, Human (HEK293, His)
Edc4
Prostanoid receptors structures, properties, and functions PMID 10508233
Rapamycin inhibits B
TATA
BU224 hydrochloride 205437
In vitro antiviral activity of the 6
A conformationally restricted guanosine analog reveals the catalytic relevance of three structures of an RNA enzyme PMID 17254949
S15176 and S16950 interaction with Cyclosporin A antiproliferative effect on cultured human lymphocytes PMID 11468012
Discovery of a First
Phospholipid metabolic adaptation promotes survival of IDH2 mutant acute myeloid leukemia cells PMID 37882467
Rivaroxaban impurity 1
Effects of uridine on the growth and differentiation of HL
Bacterial growth, detachment and cell size control on polyethylene terephthalate surfaces PMID 26464114
Fluorofenidone ameliorates cholestasis and fibrosis by inhibiting hepatic Erk/
Anaritide
DNA 聚合酶γ，催化亚基（POLG）基因
UPF
Radiation damage on Langmuir monolayers of the anionic 1.2
Concomitant Delivery of Pirarubicin and Salinomycin Synergistically Enhanced the Efficacy of Cancer Therapy and Reduced the Risk of Cancer Relapse PMID 39242397
Amino acid substitutions in the aryl hydrocarbon receptor ligand binding domain reveal YH439 as an atypical AhR activator PMID 20231332
Synthesis and quantitative structure
Piperlongumin Improves Survival in the Mouse Model of Sepsis Effect on Coagulation Factors and Lung Inflammation PMID 35831643
Ypenyl 7264
Fluorescence paper sensor meets magnetic affinity chromatography discovering potent neuraminidase inhibitors in herbal medicines PMID 39890624
Effect of magnesium on the action of oxytocin and a group of analogues on the uterus in vitro PMID 5654162
PAF1
Activation of NLRX1 by NX
N4
Discovery of a first
Galanin
Response to Programmed Cell Death
Neuropeptide Y and its C
Bronchodilating properties of the VIP receptor agonist Ro 25
GP73 reinforces cytotoxic T
Long
11
Sulfur dioxide derivatives attenuates consolidation of contextual fear memory in mice PMID 34861211
AUX1
The effects of H1
Non
Antagonists of the human adenosine A2A receptor. Part 3 Design and synthesis of pyrazolo[3,4
Cimifugin suppresses type 2 airway inflammation by binding to SPR and regulating its protein expression in a non
CCR4 mediates CCL17 (TARC)
Stn1
Changes in GABA and GABA(B) receptor expressions are involved in neuropathy in the rat cuneate nucleus following median nerve transection PMID 22290688
Development of highly potent phosphodiesterase 10A (PDE10A) inhibitors Synthesis and in vitro evaluation of 1,8
PI3K
Nuclear receptor subfamily 1 group D member 1 suppresses the proliferation, migration of adventitial fibroblasts, and vascular intimal hyperplasia via mammalian target of rapamycin complex 1/β
Dimethocaine, a synthetic cocaine derivative studies on its in vitro metabolism catalyzed by P450s and NAT2 PMID 24309420
片髓灯芯草提取物 (Juncus inflexus L.)
Bioanalysis of sulprostone, a prostaglandin E2 analogue and selective EP3 agonist, in monkey plasma by liquid chromatography
L
Cd72 Rat Pre
(2S,4S)
Cytochrome P450 1B1 contributes to increased blood pressure and cardiovascular and renal dysfunction in spontaneously hypertensive rats PMID 24477449
Substance P (free acid) adopts different conformation than native peptide in DMSO, water and DPPC bilayers PMID 11565844
The antitumor effects of an arsthinol
N
Dynamics of GLP
Inhibitory mechanism of 10
Rimegepant A Review in the Acute Treatment and Preventive Treatment of Migraine PMID 36739335
Hexocannabitriol 380495
hsa
MCE
Use of the National Surgical Quality Initiative Program in Vascular Surgery Research PMID 31344462
3
A multicenter, randomized study of argatroban versus heparin as adjunct to tissue plasminogen activator (TPA) in acute myocardial infarction myocardial infarction with novastan and TPA (MINT) study PMID 10362188
Castor1
Dehydroabietic acid 1740
Potent suppression of Kv1.3 potassium channel and IL
High
Molecular and pharmacological blockade of the EP4 receptor selectively inhibits both proliferation and invasion of human inflammatory breast cancer cells PMID 19227010
Antimicrobial agent
PanK2调节剂、基因
Metastin and its variant forms suppress migration of pancreatic cancer cells PMID 15013429
Hydrangeic acid 491
Ineffectiveness of 6,2',4'
Cirrhopetalanthrin 120090
组氨酸脱羧酶（HDC）基因
Scarb1
Discovery and Characterization of BAY
Metabolomics coupled with integrative pharmacology reveals the therapeutic effect of l
Glycolytic System in Axons Supplement Decreased ATP Levels after Axotomy of the Peripheral Nerve PMID 36894321
4
Fluoroalkane thioheterocyclic derivatives and their antitumor activity PMID 25728023
MCE
Biomimetic Peptide Nanonets Exploiting Bacterial Entrapment and Macrophage Rerousing for Combatting Infections PMID 39240217
EXP408
Dose
Synthesis and anti
BRD4 degrader
Targeting ceramide synthases for the development of new antifungals PMID 40555233
7
CXL 017
Cyclic
Antibiotic A
Phase 1 Study To Assess the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of Multiple Oral Doses of DS
Cell penetration properties of maurocalcine, a natural venom peptide active on the intracellular ryanodine receptor PMID 16545341
Mutational mapping of the transmembrane binding site of the G
Structure and Inhibitor Binding Characterization of Oncogenic MLLT1 Mutants PMID 33749253
second messenger
Liensinine alleviates high fat diet (HFD)
2
Discovery of 7, 4'
A novel lead for specific anti
Aminopyridazines as acetylcholinesterase inhibitors PMID 10052979
Selective activation of the SK1 subtype of human small
Boron
9
HDAC5 Loss Enhances Phospholipid
The neurobiology of antiepileptic drugs PMID 15208697
B
In vitro metabolism considerations, including activity testing of metabolites, in the discovery and selection of the COX
Nucleus pulposus cell
Isosorbide
Optimization of 4
Medag
Intracellular targets of moxifloxacin a comparison with other fluoroquinolones PMID 10797078
Treatment of premature labor with ritodrine a randomized controlled study PMID 379722
TRAP
Fgf22
In vitro antibacterial activity of FK041, a new orally active cephalosporin PMID 10513845
4'
Ahr
L3mbtl1
Tris
Specificity of protein kinase inhibitor peptides and induction of long
The H2S
CRBN ligand
β
CCL27 is a critical factor for the development of atopic dermatitis in the keratin
A fluorogenic probe for SNAP
DNA
Medioresinol from Eucommiae cortex improves myocardial infarction
Diarachidonin
Ku complex interacts with and stimulates the Werner protein PMID 10783163
L
Tetrahydrobiopterin 17528
Optimization of 3
Mef2d Rat Pre
Opioid receptors PMID 15189164
Bridging the gap with amide linkers rational design, synthesis, and multi
Endothelin ET(B) receptors are involved in the relaxation to the pig urinary bladder neck PMID 22460263
NAP
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