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GPR139
peptidec
Metabolic biology of 3
Synthesis and Cytotoxicity Evaluation of DOTA
Nelivaptan 439687
hepadnaviruse
MMG11
(+)
Azidoacetic Acid (2
22 6 PE
alpha
hsa
Hdac3 Mouse Pre
mmu
L
High
P2Y12 antagonist 2
Dextran sucrase (葡聚糖蔗糖酶)
β
Anti
5α
Rcan2 Rat Pre
Il27 Rat Pre
PACSIN1 Human Pre
TRAPPC8 Human Pre
ZYJ
Hdac3 Rat Pre
12
Mal
FGF20 Human Pre
Carbendazim mixture with flusilazole
hsa
2’,3’,5’
D
a
Itga2 Rat Pre
CALNN
MCE
GATA4 Human Pre
Zotadirsen
Lipoxidase, Glycine max (soybean)
5,6,7
hsa
Val
β
Mal
Anti
PROTAC BRD4 Degrader
Demethyl
Unylinker
mmu
6,7
3?
2
Insulinostatic activity of cerebellin
hsa
Dimerization quality control ensures neuronal development and survival PMID 30190310
Recent advances in the rational design and development of LIM kinase inhibitors are not enough to enter clinical trials PMID 29908439
Complement component C3a plays a critical role in endothelial activation and leukocyte recruitment into the brain PMID 26822321
4
BAY 59
Improvement of Gut Microbiota by Inhibition of P38 Mitogen
Hyodeoxycholic acid relieves neuropathic pain by activating farnesoid X receptor signaling PMID 40653266
BVT2733
N1
MC
Discovery of a novel and potent series of dianilinopyrimidineurea and urea isostere inhibitors of VEGFR2 tyrosine kinase PMID 15990302
Freezing the Bioactive Conformation to Boost Potency The Identification of BAY 85
Plasma membrane isolation using immobilized concanavalin A magnetic beads PMID 22903707
IGFBP3 enhances adipose
SRD5A2 抗体 (YA3540)（SRD5A2 Antibody (YA3540)）
First non
Steroidal saponins from fresh stem of Dracaena cochinchinensis PMID 15013689
Neuropeptide SF(mouse,rat) TFA
Casopitant 414910
Structure
Discovery of disubstituted xylylene derivatives as small molecule direct inhibitors of Keap1
Fmoc
KG
Maximin8
EOS
Placental Fatty Acid Metabolism and Transport in a Rat Model of Gestational Diabetes Mellitus PMID 37288271
Knockdown of SGK1 alleviates the IL
TLR4
PLLA10000
Pinostilbenoside
thallium
3,4
Development of an intranasal formulation containing indomethacin and xylometazoline for rhinosinusitis treatment PMID 36524913
NDSB 256
BGG463 890129
3
GSK190937 2651234
Hippo
An L
BGE
Anticancer properties of indole derivatives as IsoCombretastatin A
Betahistine mesylate 54856
gonads
Osutidine
ion indicator
Platyphylloside 90803
IL11
WAY
Hericene A 157207
AMI
Nrf2
The discovery of I
Analysis of ginsenosides in Panax ginseng in high pressure microwave
ATB337
New transition metal ion complexes with benzimidazole
A novel diamino
Comprehensive analysis of nonsurrounded nucleolus and surrounded nucleolus oocytes on chromatin accessibility using ATAC
ETH5294
Structure guided design of potent indole
PT150 189035
Surface expression of PEDV nucleocapsid protein facilitates NK cell
Altafur
ferment
Fenchone 1195
Isolation and characterization of a new cytotoxic dihydrophenanthrene from Dioscorea membranacea rhizomes and its activity against five human cancer cell lines PMID 25149021
The K252a derivatives, inhibitors for the PAK/MLK kinase family selectively block the growth of RAS transformants PMID 12184411
The endonuclease IV family of apurinic/apyrimidinic endonucleases PMID 20667510
CR
IRAK
Synthesis and biological evaluation of imidamide analogs as selective anti
Gliclazide 21187
Cytotoxic effects of sinococuline PMID 8616827
The selective SYK inhibitor P505
Farrerol directly activates the deubiqutinase UCHL3 to promote DNA repair and reprogramming when mediated by somatic cell nuclear transfer PMID 37012254
Toward chelerythrine optimization Analogues designed by molecular simplification exhibit selective growth inhibition in non
Identification of Potent and Selective RIPK2 Inhibitors for the Treatment of Inflammatory Diseases PMID 29057049
2
PD153035, a tyrosine kinase inhibitor, prevents epidermal growth factor receptor activation and inhibits growth of cancer cells in a receptor number
Prediction of Synergistic Drug Combinations for Prostate Cancer by Transcriptomic and Network Characteristics PMID 33986671
urchin
Design and Application of Cereblon
Fat mass and obesity
Discovery of a small
A
Alternative Hapten Design for Zearalenone Immunoreagent Generation PMID 35324682
Dabcyl acid 6268
Synthesis and antiviral activity of new acrylamide derivatives containing 1,2,3
Luciferase
Erythropoietic protoporphyria. A new porphyria syndrome with solar urticaria due to protoporphyrinaemia PMID 13765301
Selective Glucocorticoid Receptor Modulators (SGRMs) Delay Castrate
Coronarin D Me ether
IND71677
α
The polycomb group protein enhancer of zeste 2 is a novel therapeutic target for cervical cancer PMID 25739318
[Pharmacotherapy
DB1976 dihydrochloride 2369663
Using chimeric mice with humanized livers to predict human drug metabolism and a drug
A novel mitochondriotoxic small molecule that selectively inhibits tumor cell growth PMID 12150823
First
Biotinylated probes for in situ hybridization histochemistry use for mRNA detection PMID 8245422
Matrix stiffness
Big CHAP 86303
COVID
An examination of the euphorbiaceae of Hong Kong. VI. Isolation and structure of glochidonol, a new triterpene ketol from Glochidion wrightii Benth PMID 5817977
Type I phosphatidylinositol 4
27
Glial expression of Drosophila UBE3A causes spontaneous seizures that can be modulated by 5
CL
Hypericin Nanoparticles
Nucleoside Analogs Radiosensitize G0 Cells by Activating DNA End Resection and Alternative End
Discovery of Thieno[2,3
Lupane and 18α
Demethoxyencecalin 19013
CDP 571
Heat shock protein 70 inhibitors suppress androgen receptor expression in LNCaP95 prostate cancer cells PMID 28691182
A newly developed PLD1 inhibitor ameliorates rheumatoid arthritis by regulating pathogenic T and B cells and inhibiting osteoclast differentiation PMID 37722567
TLR2
Crystal structure of the HhaI DNA methyltransferase complexed with S
The search for potent, small molecule NNRTIs A review PMID 19632850
Baicalin prevents fibrosis of human trabecular meshwork cells via inhibiting the MyD88/NF
Tiagabine 115103
TH5487 specifically targets NLRP3 in FCAS patients resistant to MCC950 PMID 40661406
Comparative Analysis of Small
ARVs
Rationale and design for the development of a novel nitroxyl donor in patients with acute heart failure PMID 31168885
PLX
BCX4430, a novel nucleoside analog, effectively treats yellow fever in a Hamster model PMID 25155605
Rubitecan 9
cPLA2α
Hypo
AalphaC
3
Effects of the antitussive drug cloperastine on ventricular repolarization in halothane
Design, synthesis and optimization of bis
N
Piperoxan hydrochloride (Standard) (盐酸哌罗克生 (标准品))
Nur77 modulator 1 2469975
The alpha1
CGP52421
GS6201
Characterization of a dual BET/HDAC inhibitor for treatment of pancreatic ductal adenocarcinoma PMID 32599645
Examination of Effective Buccal Absorption of Salmon Calcitonin Using Cell
Human Growth Hormone (1
Ergocalciferol and cholecalciferol in CKD PMID 22560832
Geldanamycin derivatives and neuroprotective effect on cultured P19
Metabolism, excretion, and pharmacokinetics of ((3,3
Antitumor effects of immunotoxins are enhanced by lowering HCK or treatment with SRC kinase inhibitors PMID 24145282
Inhibition of the C1s Protease and the Classical Complement Pathway by 6
Detailed analysis of cortisol, cortisone and their tetrahydro
Silence of linc00023 inhibits pyroptosis and promotes cell proliferation via regulating p53 PMID 37429368
The novel dipeptidyl peptidase
lethal sepsis
Agonist and antagonist activities on human NPFF(2) receptors of the NPY ligands GR231118 and BIBP3226 PMID 11325787
RAB31 Human Pre
In vitro and in vivo characterization of SARS
Hydrazyl hydroxycoumarins as new potential conquerors towards Pseudomonas aeruginosa PMID 38494040
EAC3I 209004
AMG
2
MAP3K4 promotes fetal and placental growth by controlling the receptor tyrosine kinases IGF1R/IR and Akt signaling pathway PMID 35921893
Cilia locally synthesize proteins to sustain their ultrastructure and functions PMID 34848703
Acetic acid
Agranulocytosis after consumption of cocaine adulterated with levamisole PMID 19153405
Pharmacological profile of LF 16
PRMT5
Evogliptin a new dipeptidyl peptidase inhibitor for the treatment of type 2 diabetes PMID 27156529
Gα Protein Mediates High
The effect of isosaponarin isolated from wasabi leaf on collagen synthesis in human fibroblasts and its underlying mechanism PMID 20349148
Gut microbiota
Melperone but not bisoprolol or metoprolol is a clinically relevant inhibitor of CYP2D6 evidence from a therapeutic drug monitoring survey PMID 25940834
DC07090 879070
OCS
Agnuside 11027
Construction and evaluation of BSA
5
Neuronal CCL2 is upregulated during hepatic encephalopathy and contributes to microglia activation and neurological decline PMID 25012628
Synthesis of CDDO
Potent inhibition of human liver aldehyde oxidase by raloxifene PMID 14709625
Norflurazon 27314
Diaryl hydroxylamines as pan or dual inhibitors of indoleamine 2,3
Isolation of novel cell
Diversity of mitochondria
Tryptamine
Real
The inhibitory effect of enfenamic acid (Tromaril) on hepatic gluconeogenesis in Swiss albino mice PMID 3004495
A new idea for simple and rapid monitoring of gene expression requirement of nucleotide sequences encoding an N
Targeting Dlat
Cyantraniliprole impairs reproductive parameters by inducing oxidative stress in adult female wistar rats PMID 34968715
Agaridoxin 58298
Carbadox 6804
Design, synthesis, and biological evaluation of ligustrazine
The tick saliva peptide HIDfsin2 promotes the tick
8
EphA2 signaling is impacted by carcinoembryonic antigen cell adhesion molecule 1
Novel arylsulfonamide derivatives with 5
ETA receptor antagonists inhibit intimal smooth muscle cell proliferation in human vessels PMID 12193082
CD11c 抗体（CD11c Antibody）
Synthetic small molecule furin inhibitors derived from 2,5
The prevention of encephalitis due to the viruses of eastern equine encephalomyelitis and louping
A Novel Viral Assembly Inhibitor Blocks SARS
Methyl heptadecanoate 1731
3beta
Pramipexole improves depression
Differential metabolic responses of Beauveria bassiana cultured in pupae extracts, root exudates and its interactions with insect and plant PMID 25584432
Vipadenant 442908
Up
Daraxonrasib, a pan
Identification of antiviral compounds against equid herpesvirus
PK11000 38275
Dihydroberberine 483
Gastrodin protects against high glucose
Acarviosin 80943
Luvagrobart
Calebin A 336784
Effects of etifoxine on ligand binding to GABA(A) receptors in rodents PMID 12354631
High
RGB286147
DP2 antagonist
Fuberidazole
dTTPαS 18883
Glul Rat Pre
UNC5H2
PW0464
Antithrombotic effects of the prostacyclin analogue naxaprostene after oral and intraduodenal application in rabbit carotid artery thrombosis PMID 1632291
AMPA receptor modulator
Ro 01
KPRP Human Pre
Kmeriol and other aromatic constituents of Kmeria duperreana PMID 2798315
Function, activity, and membrane targeting of cytosolic phospholipase A(2)zeta in mouse lung fibroblasts PMID 17293613
γ
Ramos cels
Investigation of intracellular magnesium mobilization pathways I PC12 cells B simultaneous Mg
Phlda1 Rat Pre
DW 34
NSC258308
Mechanism of Herbicidal Action and Rice Selectivity of Iptriazopyrid A Novel Azole Carboxamide
ATH3G10
BMP
Taraxasterol acetate targets RNF31 to inhibit RNF31/p53 axis
microtubule structure
The synergic modeling for the binding of fluoroquinolone antibiotics to the hERG potassium channel PMID 23711922
CB65
RG 6866 120602
Progress of bis(heteroaryl)piperazines (BHAPs) as non
Fluorocyclopentenyl
Benzodiazepines
Xanthamide
CC
Topical N
Synergy of 5
Porphyrin
The Discovery of GS
Mivacurium dichloride 106861
Pellotine
MSI1 Human Pre
Exacerbated ischemia
Timapiprant 851723
The receptor for advanced glycation end products is required for β
CIM0216 1031496
Design, synthesis and biological evaluation of thiazolyl
NSC288020
MCE
[Neocodion misuse evolution between 1992 and 2002] PMID 15648308
SCO
ApoE In Vitro Studies of a Small Molecule Effector PMID 27065061
Inhibitory effect of rhetsinine isolated from Evodia rutaecarpa on aldose reductase activity PMID 17498942
F
ELF5
CbZ
PI3Kγδ inhibition suppresses key disease features in a rat model of asthma PMID 38654248
HCV NS5B polymerase
Hatomamicin 116290
Casein kinase 2 is essential for mitophagy PMID 23897086
CP 461 227619
Dimethyl suberimidate dihydrochloride 34490
LC
RNF5
A Trimethoprim Conjugate of Thiomaltose Has Enhanced Antibacterial Efficacy In Vivo PMID 29660287
C18
P
Azaribine 2169
BML 277
Loganin protects against myocardial ischemia
Chemical Stability of Plerixafor after Opening of Single
W2476 represses TXNIP transcription via dephosphorylation of FOXO1 at Ser319 PMID 33560565
Chemical constituents from Inonotus obliquus and their biological activities PMID 24359303
Tiospirone hydrochloride 87691
Isolation, Antimicrobial Susceptibility, and Genotypes of Three Pasteurellaeae Species Prevalent on Pig Farms in China Between 2021 and 2023 PMID 40284774
NFAT1 Signaling Contributes to Bone Cancer Pain by Regulating IL
SOS1/KRAS
Using SV119
Brain
Thioxanthenone
PTPN3 Human Pre
Theabrownins improve burn
Synthetic Essentiality of Tryptophan 2,3
HepArrest
Apelin
Biological activities of fusarochromanone a potent anti
Methyl dodonate A acetate
Eps15 Rat Pre
TP53AIP1 Human Pre
Azadirachtin D
GnRH
ATX inhibitor 24
TIRAP Human Pre
MIF Human Pre
TAP2 Human Pre
Xpo7 Mouse Pre
IL22RA1 Human Pre
hsa
SARS
Bisindolylmaleimide X (BIM
mmu
hsa
3
Bicyclo
PPP1CC 蛋白, Human (His)
MCE
hsa
Yellow brown XF
S100A5 蛋白, Mouse (His)
ITSA
Mal
AGTRAP Human Pre
C16 Cy5 SM chloride
WT
FBXO21 Human Pre
苦乐果提取物 (Garcinia kola Heckel)
4
MCE
hsa
Gm2a
Maresin1 ameliorates ventricular remodelling and arrhythmia in mice models of myocardial infarction via NRF2/HO
Hippuric acid
Taxus cuspidata
GMNN
1
Discovery and structure
Discovery of (quinazolin
Biological activity and chemistry of taxoids from the Japanese yew, Taxus cuspidata PMID 14987066
MAN2B1 Human Pre
G protein
Purification, characterization and bioactivities of polysaccharides from Pleurotus ferulae PMID 28436508
Cyclization
DKM 2
The design and synthesis of human branched
Novel, broad
GLP
DPP
Heme
Rhapontisterone 137476
Fibrostatin A 91776
Acetylcholinesterase inhibitors from the roots of Angelica dahurica PMID 12510838
AZD
Structural and Biosynthetic Analysis of the Fabrubactins, Unusual Siderophores from Agrobacterium fabrum Strain C58 PMID 33373180
Phenibut
Effect of norbinaltorphimine on ∆⁹
BNN
Circumdatin A, B, and C Three New Benzodiazepine Alkaloids Isolated from a Culture of the Fungus Aspergillus ochraceus PMID 11674237
Fadaltran 1799809
Desfluoro
A first generation inhibitor of human Greatwall kinase, enabled by structural and functional characterisation of a minimal kinase domain construct PMID 27563826
UV
AHMT 1750
Histamine Intolerance Originates in the Gut PMID 33921522
热休克转录因子 1（Hsf1）基因
Regaloside H
Viridicatin
GSK2807
MMAE
Antitumor agent
Fkbp2
Toonaciliatin M 93930
Aurachin C
Nopol
TAP311
EP5
Inhibition of human skin fibroblast collagenase, thermolysin, and Pseudomonas aeruginosa elastase by peptide hydroxamic acids PMID 1322694
Degradation and inhibition of epigenetic regulatory protein BRD4 exacerbate Alzheimer's disease
Highly Efficient Thiol
EML4
Potential Therapeutic Agents for Feline Calicivirus Infection PMID 30115859
GLS1 Inhibitor
Pyrazole ligands structure
acinetobacter baumannii
MCE
Pharmacokinetics and pharmacodynamics of sibrafiban alone or in combination with ticlopidine and aspirin PMID 10718778
TMAO promotes apoptosis and oxidative stress of pancreatic acinar cells by mediating IRE1α
PSIP1 Human Pre
HF
Biotransformation of pantoprazole by the fungus Cunninghamella blakesleeana PMID 16012078
BCL
GS8588
Naphthofluorescein 61419
Novel alpha
Echinocandin B 54651
GSK
Mensacarcin 808750
Investigation of In
Anti
Con B 1
PDE4D7
MC3482
Fucose biosynthesis and biological function in mammals PMID 12651883
A novel compound RS
Caspase
In vitro evaluation of secoiridoid glucosides from the fruits of Ligustrum lucidum as antiviral agents PMID 11724241
BET
CendR
AMG
SDZ 220
Methyl 2α
Discovery of potent and orally bioavailable inhibitors of Human Uric Acid Transporter 1 (hURAT1) and binding mode prediction using homology model PMID 26704267
Cytotoxicity of labdane
Targeting CCR3 with antagonist SB 328437 sensitizes 5‑fluorouracil‑resistant gastric cancer cells Experimental evidence and computational insights PMID 38737977
Triterpenoids with neurotrophic activity from Ganoderma lucidum PMID 21671206
DMU
BAT6026, a novel anti
Nickel(II) oxide 1313
14862
TRP
ATH686 853299
LH
MEK4
Targeting voltage
Jasmoside
Clinical pharmacological innovation in the treatment of depression PMID 37000975
Phenotypic Hit Identification and Optimization of Novel Pan
OT
Parkinson disease related ATP13A2 evolved early in animal evolution PMID 29505581
The degree of esterification influences the bioactivity of pectic polysaccharides isolated from Lithocarpus litseifolius PMID 40297662
Dkc1 Rat Pre
Tolciclate 50838
OVA
4,5
N
BC05
Pygenic Acid A (PA) Sensitizes Metastatic Breast Cancer Cells to Anoikis and Inhibits Metastasis In Vivo PMID 33182770
Benastatin B 138968
GSK199
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