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IL7R Human Pre
(S)
SCH
Etevritamab 2329692
Bax 抗体 (YA6207)（Bax Antibody (YA6207)）
Drd3 Mouse Pre
GPX4 activator 2
2
cadaverine
EtOH
Ramatroban
IACS010759
ZY 444
spectrometry
Elane
Detailed characterisation of the trypanosome nuclear pore architecture reveals conserved asymmetrical functional hubs that drive mRNA export PMID 39899609
7
N
GBR
(
UCM765 944284
thiolysis
Senecivernine 72755
Purified complement C3b triggers phagocytosis and activation of human neutrophils via complement receptor 1 PMID 36609665
Histone H3 (acetyl K27) 抗体 (YA735)（Histone H3 (acetyl K27) Antibody (YA735)）
Discovery of 6,7
Structure
RAB7 activity is required for the regulation of mitophagy in oocyte meiosis and oocyte quality control during ovarian aging PMID 34229552
l
Natural product
Isoguvacine binding, uptake, and release relation to the GABA system PMID 6854327
Site
Regulation and function of MeCP2 Ser421 phosphorylation in U50488
GSK317354A 874119
Identification of small molecule activators targeting TYK2 pseudokinase domain PMID 40209917
In Vitro Metabolite Formation in Human Hepatocytes and Cardiomyocytes and Metabolism and Tissue Distribution in Monkeys of the 2'
The IL
The mGluR5 positive allosteric modulator CDPPB inhibits SO₂
The inhibitory effect and targets of CRM197 on tumor growth in arsenic
Eradication of Central Nervous System Leukemia of T
Propranolol Activates the Orphan Nuclear Receptor TLX to Counteract Proliferation and Migration of Glioblastoma Cells PMID 34115934
Discovery of a DNA Topoisomerase I Inhibitor Huanglongmycin N and Its Congeners from Streptomyces sp. CB09001 PMID 34709824
Carbenoxolone
BacFlash signals acid
Role of interferon
CD63
Mycobacterial tuberculosis
NSD
Mal
Linalool
6
MK
Development and investigation of a QuEChERS
U
Elcatonin
Metallo
Desmethylene paroxetine hydrochloride 1394861
6'
LVGN
GS 5290
U62066
N
Engeletin
SQ
ACT 678689
Spautin
RXDX 106
XmAb14045
Insulinase
Comparative analysis of B7
PAMP
Carbon monoxide attenuates cellular senescence
B4galt1 Mouse Pre
8
4108
Chemogenetic Approaches to Explore the Functions of Free Fatty Acid Receptor 2 PMID 33495026
GDF6 Human Pre
Phenylbutazone in the horse a review PMID 3517382
A chemical compound that stimulates the human homologous recombination protein RAD51 PMID 18840682
Isoprenylated Flavonoids with PTP1B Inhibition from Macaranga denticulata PMID 26791751
基质金属肽酶 26（MMP26）基因
Genetic Analysis of JNK MAPK Signaling in Stress
Prostate
Preclinical evaluation of terbinafine in vivo PMID 2598485
Pharmacology of human sulphonylurea receptor SUR1 and inward rectifier K(+) channel Kir6.2 combination expressed in HEK
Hepatic FcRn regulates albumin homeostasis and susceptibility to liver injury PMID 28330995
GNE
Liver abscess induced by intestinal hypervirulent Klebsiella pneumoniae through down
Membrane
Nicaraven attenuates radiation
Salvianolic acid B alleviates diabetic endothelial and mitochondrial dysfunction by down
Expression of an interleukin
Involvement of ferroptosis in eribulin
Synthesis and anti
Guanidine
Regulation of myometrial contraction by ATP
TACI 抗体 (YA1385)（TACI Antibody (YA1385)）
Alleviation of mechanical and thermal allodynia by CGRP(8
Biotinylated Stealth magnetoliposomes PMID 12426077
Broad sensitivity of rodent arrhythmia models to class I, II, III, and IV antiarrhythmic agents PMID 2726785
Design, synthesis and apoptosis
Trpc1
Synthesis of mitochondria
DNAM
Chemogenomic screening identifies the Hsp70 co
Anti
PSCA 蛋白, Mouse (HEK293, His)
DCTN1 蛋白, Human (His
Self
Differential effects of histamine H(3) receptor inverse agonist thioperamide, given alone or in combination with the N
MCE
Adriforant 943057
Exploring new near
Inhibition of LpxC Increases Antibiotic Susceptibility in Acinetobacter baumannii PMID 27270288
Synthesis and biological evaluation of 3,4,6
A mast cell receptor mediates post
Optimization of 3
Antiangiogenic effect of dual/selective alpha(5)beta(1)/alpha(v)beta(3) integrin antagonists designed on partially modified retro
PTEN counteracts FBXL2 to promote IP3R3
CD00509 27430
Synergistic efficacy of Bisbenzimidazole and Carbonyl Cyanide 3
COX
Self
Comparative analysis and directed protein evolution yield an improved degron technology with minimal basal degradation, rapid inducible depletion, and faster recovery of target proteins PMID 39606491
Analogs of FTY720 inhibit TRPM7 but not S1PRs and exert multimodal anti
Ponatinib
Synthesis of 3
Effects of gamma
FGFR1 抗体 (YA441)（FGFR1 Antibody (YA441)）
DS
A human ICAM
9
Antagonistic effects of antimuscarinic drugs on alpha 1
Treatment of anemia with microencapsulated ferrous fumarate plus ascorbic acid supplied as sprinkles to complementary (weaning) foods PMID 11722961
Programmable alignment media from self
Chemokine CXCL10/CXCR3 signaling contributes to neuropathic pain in spinal cord and dorsal root ganglia after chronic constriction injury in rats PMID 30448292
Prevention of aspirin
Histone H3 (acetyl K14) 抗体 (YA375)（Histone H3 (acetyl K14) Antibody (YA375)）
Alectinib analog 1256577
GSK1790627 871701
Fosfomycin Pharmacological, Clinical and Future Perspectives PMID 29088073
Quantitative Analysis of Benzyl Isothiocyanate in Salvadora persica Extract and Dental Care Herbal Formulations Using Reversed Phase C18 High
Deciphering the Therapeutic Potential of Novel Pentyloxyamide
The Caulobacter crescentus FlbD protein acts at ftr sequence elements both to activate and to repress transcription of cell cycle
84060
(S,S)
Two New Succinimide Derivatives Cladosporitins A and B from the Mangrove
Toxicologic study of carboxyatractyloside (active principle in cocklebur
5
Endothelin
A novel selective positive allosteric modulator of metabotropic glutamate receptor subtype 5 has in vivo activity and antipsychotic
pro
Timcevibart 2857862
NSD
Synthesis and antiviral activity of thiazolyl hydrazones against dengue virus PMID 41077226
Design, synthesis, and biological evaluation of 14
CUMS
CDT1 抗体 (YA507)（CDT1 Antibody (YA507)）
Dnmt1 抗体 (YA476)（Dnmt1 Antibody (YA476)）
Anthranilyl
(Z)
Linifanib
A new mechanism of 6
Monoethylglycinexylidide
Analgesic effect of sinomenine in rodents after inflammation and nerve injury PMID 24120369
OSS_128167 887686
New steroid acids from Antrodia cinnamomea, a fungal parasite of Cinnamomum micranthum PMID 8594142
Kcna3
8347
Recent advances in the development of selective human MAO
Antagonism of CXCR3 inhibits lung metastasis in a murine model of metastatic breast cancer PMID 16885372
MCE
Evidence that CYP2C19 is the major (S)
PtdIns
Surface Modification of Polymeric Nanoparticles with M2pep Peptide for Drug Delivery to Tumor
Dibenzo[b,e][1,4]dioxin
HCV
AhR modulator
Effect of iprodione, a dicarboximide fungicide, on primary cultured rainbow trout (Oncorhynchus mykiss) hepatocytes PMID 11451425
Cytotoxic and antimalarial constituents of the roots of Eurycoma longifolia PMID 1800638
Increased arylhydrocarbon receptor expression offers a potential therapeutic target for pancreatic cancer PMID 12203118
MCE
hsa
Fibroblast growth factor 21 corrects obesity in mice PMID 18687777
Methotrexate
LC
DK419
Interaction of N
hsa
CCI52 sensitizes tumors to 6
GW274150 and GW273629 are potent and highly selective inhibitors of inducible nitric oxide synthase in vitro and in vivo PMID 15778742
D
Bis(dibenzylideneacetone)palladium 32005
Poly
EN4 1197824
JTP
Ferfluor1
Influenza Matrix Protein (61
6
AMG 487 473719
Quaternary heterocyclylamino beta
Poly
Innovative therapies for acute bacterial skin and skin
A high
The ameliorating effects of stigmasterol on scopolamine
S
5
SH3GL1 抗体 (YA4456)（SH3GL1 Antibody (YA4456)）
氯索洛芬
fruit sugar
Interaction of zalcitabine with human organic anion transporter 1 PMID 16724555
Nepetalactone content and antibacterial activity of the essential oils from different parts of Nepeta persica PMID 20433086
A prospective, randomized, controlled, exploratory study of comprehensive dietary advice in ulcerative colitis impact on disease activity and quality of life PMID 24942954
Acetylcholinesterase complexes with the natural product inhibitors dihydrotanshinone I and territrem B binding site assignment from inhibitor competition and validation through crystal structure determination PMID 24573600
Psmd2 Rat Pre
Concanavalin A
An insight on medicinal attributes of 1,2,4
Tefluthrin 79538
Chelidonine Induces Caspase
Tunicamycin
Macrocyclic pyrrolizidine alkaloids from Senecio anonymus. Separation of a complex alkaloid extract using droplet counter
CBX7 Human Pre
Vitamin D
AP 24534
NF157 104869
A role for MAP kinase signaling in behavioral models of depression and antidepressant treatment PMID 16945347
Lgals4
Sphinganine recruits TLR4 adaptors in macrophages and promotes inflammation in murine models of sepsis and melanoma PMID 39025856
Use of oral fluconazole during pregnancy and the risk of birth defects PMID 23984730
Furin Substrate 174838
PDLHB (MW 30000
Strychnos nux
Discovery of novel orally bioavailable oxaborole 6
The structure
Synthesis, antibacterial and antifungal activity of new 3
In vitro and in silico evaluation of inhibitory effects of bisphenol derivatives on acetylcholinesterase of electric eel (Electrophorus electricus L.) PMID 35843445
Promotion of Arabidopsis immune responses by a rhizosphere fungus via supply of pipecolic acid to plants and selective augment of phytoalexins PMID 36449213
B4GALT1 Human Pre
p
HDAC6
Synthesis of novel estrogen receptor antagonists using metal
Rational design, synthesis, antiproliferative activity against MCF
2,4
Cucurbitacins are insect steroid hormone antagonists acting at the ecdysteroid receptor PMID 9581538
BSA reduces inhibition in a TaqMan assay for the detection of Batrachochytrium dendrobatidis PMID 21268973
Design and synthesis of 1,3
GALT 抗体 (YA2925)（GALT Antibody (YA2925)）
7,8
hydrolysis
N6
GSPT1 degrader
Investigation of (E)
Role of local bioactivation of vitamin D by CYP27A1 and CYP2R1 in the control of cell growth in normal endometrium and endometrial carcinoma PMID 24732451
Metal
Synthesis and evaluation of hydrophilic linkers for antibody
α
A
Gastric Cancer Cell
Laptm5
CD46 分子（CD46）基因
MCE
Rbm15
Peripheral and central administration of xenin and neurotensin suppress food intake in rodents PMID 19214175
PMED
Isoremoxipride 107188
TUBGCP4 Human Pre
Effects of zamicastat treatment in a genetic model of salt
Ebselen oxide 104473
AP
Inocoterone and acne. The effect of a topical antiandrogen results of a multicenter clinical trial PMID 1387778
A novel free radical scavenger, nicaraven, inhibits human platelet aggregation in vitro PMID 10047928
TGF
Specialization among iron
TRPV4 inhibition counteracts edema and inflammation and improves pulmonary function and oxygen saturation in chemically induced acute lung injury PMID 24838754
DPHC From Alpinia officinarum Ameliorates Oxidative Stress and Insulin Resistance via Activation of Nrf2/ARE Pathway in db/db Mice and High Glucose
The melanocortin ACTH 1
GW274150 dihydrochloride 438542
A selective inducible NOS dimerization inhibitor prevents systemic, cardiac, and pulmonary hemodynamic dysfunction in endotoxemic mice PMID 12907425
Structure
Measurement of technetium
Foenumoside B from Lysimachia foenum
G721
E2F 转录因子 8（E2F8）基因
Nf1
Hedgehog inhibitors from Artocarpus communis and Hyptis suaveolens PMID 26178912
NRF1 knockdown alleviates lipopolysaccharide
Adrenic acid metabolites as endogenous endothelium
Small molecule Plasmodium FKBP35 inhibitor as a potential antimalaria agent PMID 23974147
Oligomycin E, a new antitumor antibiotic produced by Streptomyces sp. MCI
Fmoc
Neurochemical changes underlying cognitive impairment in olfactory bulbectomized rats and the impact of the mGlu5
Prdm12 governs an epigenetic checkpoint linking neuroimmune cross
Epigomisin O 73036
AL 39324
Five new diprenylated flavonols from the leaves of Broussonetia kazinoki PMID 11575957
Ponatinib 943319
Chronic Glucocorticoid Exposure Induced a S1PR2
VCAM
An assay for sphingosine kinase activity using biotinylated sphingosine and streptavidin
Current advances of small molecule E3 ligands for proteolysis
Activity of 2
BMS
Gut microbial DL
N,N'
Transcriptomics changes of calcitonin gene
Discovery of novel biphenyl compounds bearing hydroxamic acid moiety as the first PD
Hyou1 Rat Pre
Phospholipase D PMID 15052340
Boc
Retn
OncomiR
CHI3L1
Discovery of an autoinhibited conformation in mesotrypsin reveals a strategy for selective serine protease inhibition PMID 40614191
CGRP Receptor
OS
COX
Molecular determinants of substrate and inhibitor specificities of the Penicillium griseofulvum family 11 xylanases PMID 19118652
Dtnb
Discovery of novel carboxylesterase 2 inhibitors for the treatment of delayed diarrhea and ulcerative colitis PMID 37567318
A4galt Rat Pre
PA (224
Synthesis and biological evaluation of 4
DEL
Inositol 1,3,4,5
SH
RS
Inhibition of AKR1B10
Identification of DK419, a potent inhibitor of Wnt/β
Discovery of novel ENPP1 inhibitors with benzotriazole core for cancer immunotherapy PMID 41687265
CTLA
Context
Choline alphoscerate (alpha
Hypoxia
Preclinical pharmacokinetics and in vitro metabolism of BMS
Transporter
DK 419
4,4& 039;
Endocrine regulation of energy metabolism by the skeleton PMID 17693256
A phase I trial of PRN1008, a novel reversible covalent inhibitor of Bruton's tyrosine kinase, in healthy volunteers PMID 28636208
Methylenecyclopropylpyruvate 5746
8
Discovery of 4
2',5'
stroke
CTLA
DiMethyl
Eif5a
Novel nonsecosteroidal vitamin D receptor modulator inhibits the growth of LNCaP xenograft tumors in athymic mice without increased serum calcium PMID 11746268
N
CGRP (83
Transcriptional function of E2A, Ebf1, Pax5, Ikaros and Aiolos analyzed by in vivo acute protein degradation in early B cell development PMID 39179932
CML With Mutant ASXL1 Showed Decreased Sensitivity to TKI Treatment via Upregulation of the ALOX5
Atrial natriuretic factor (1
G721
3’,5’
ADC Linker
Structure
Calcium
Phosphatase
KER047 succinate 2416307
Expression and role of MIG/CXCR3 axis in mantle cell lymphoma PMID 33197439
Design, synthesis and anticancer properties of novel oxa/azaspiro[4,5]trienones as potent apoptosis inducers through mitochondrial disruption PMID 26163220
Mat2b
Lack of significant modifying effect of arctiin on prostate carcinogenesis in probasin/SV40 T antigen transgenic rats PMID 15863263
Discovery of 3
Hes1 upregulation contributes to the development of FIP1L1
hsa
STK38 Human Pre
N
Sedolisins, a new class of secreted proteases from Aspergillus fumigatus with endoprotease or tripeptidyl
Cytotoxic activity, apoptosis induction and structure
A cell
Stimulatory effect of romurtide on hematopoiesis in monkeys PMID 2049113
Inhibition of Simian Virus 40 replication by targeting the molecular chaperone function and ATPase activity of T antigen PMID 19200446
Effects of GW274150, a novel and selective inhibitor of iNOS activity, in acute lung inflammation PMID 14769784
Influenza A virus
Neuropeptide apelin presented in the dopaminergic neurons modulates the neuronal excitability in the substantia nigra pars compacta PMID 36041497
Concanavalin A
帕拉替尼
ENPP5 抗体 (YA6554)（ENPP5 Antibody (YA6554)）
G721
Discovery and Development of N
Design, synthesis, and anti
β
Retn Rat Pre
泊那替尼
G721
1,2
(2S)
CRBN ligand250
Structure
4,4'
CTLA
Discovery of Potent Antiallergic Agents Based on an o
A family of tissue
Sinomenine ester derivative inhibits glioblastoma by inducing mitochondria
iron
Stigmasta
8
Dram1 Rat Pre
LCB 03
N
D
N
Sofpironium Bromide First Approval PMID 33236266
Conversion of human fibroblasts into functional cardiomyocytes by small molecules PMID 27127239
Osbond acid 25182
A
Barzolvolimab 2438203
Rilzabrutinib 1575596
Effectors of HIV
(R)
Targeting BRCA1
Silica
Actions and addiction liabilities of alpha
1,2
Anisodine 52646
Hypermongones A
The murine version of BAN2401 (mAb158) selectively reduces amyloid
ETH 157 61595
Cellular prion protein is released on exosomes from activated platelets PMID 16434486
Bile acids inhibit cholinergic constriction in proximal and peripheral airways from humans and rodents PMID 31800261
Chelerythrine 34316
Selective functional inhibition of JAK
Methacrylic acid N
GLP
HBV
Histone H3 (acetyl K18) 抗体 (YA736)（Histone H3 (acetyl K18) Antibody (YA736)）
BBOX1 restrains TBK1
L17E
(R)
1,4
EED226 2083627
L
Reduction of human monocytic cell neurotoxicity and cytokine secretion by ligands of the cannabinoid
MK 1029
Malonylcarnitine in newborns with non
Bersanlimab 1987854
A High
Wilforine
HS
Concordant but Varied Phenotypes among Duchenne Muscular Dystrophy Patient
Cd80
hsa
RPR 208707
Mapping the binding site of tissue kallikrein preparation and testing of all possible substrate analog inhibitors homologous with the sequence of kininogen between Ser386 and Gln392 PMID 1507198
UR
Catestatin 142211
Cyb5r3
Muzolimine
BCX 1470 217099
Nitric Oxide
Mdh2
Taplitumomab
Insecticidal agent 27
XR
Surfactin C1
hsa
SHMT
Protective effect of esculentoside A on lipopolysaccharide
Torutamig
JAK1 Inhibition Blocks Lethal Immune Hypersensitivity in a Mouse Model of Down Syndrome PMID 33207208
Dynapyrazole
DePARylation is critical for S phase progression and cell survival PMID 38578205
hsa
SU 0383
Boerhaavia diffusa
Mal
HDAC6
NNMTi 42464
BIVV
M1
Bz
2
PF
FNTA Human Pre
ICMT
mutant IDH1
An auxin
URB937
twitching motility
Ten
N
GSK 9772
mmu
YM14673
Aminooxy
XY028
Autophagy
Sftpb Mouse Pre
Astragenol
WP 1193
GSK040 2752331
Cyclooctyne
CYT0851
1
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