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Pyridinolcarbamate and experimental atherosclerosis. Correlation of hypocholesterolemic and antiatherogenic effects PMID 728238
(R)
Suppression of PAPP
DYRKs
MCE
57335
HBV
Cevidoplenib 1703788
The unexpected role of lymphotoxin beta receptor signaling in carcinogenesis from lymphoid tissue formation to liver and prostate cancer development PMID 20603617
Genipin stabilized fibrin microbeads Carrying cytokines to form niches for stem cell differentiation PMID 40391599
IL
(R)
4
Ozanezumab 1310680
Identification of the HPV
Fat1
3
STAT3
Theranostic Agents for Photodynamic Therapy of Prostate Cancer by Targeting Prostate
MS275 Inhibits Neuroblastoma Cell Growth by Mediating H3K27ac/PROX1 Axis In Silico and In Vitro PMID 40601211
SLC1A1 Human Pre
Regulation of T cell activation and tolerance by PDL2 PMID 16864790
Exploring the interaction between human focal adhesion kinase and inhibitors a molecular dynamic simulation and free energy calculations PMID 26549408
Rhodanine a selective inhibitor of the multiplication of echovirus 12 PMID 4982794
Endocytosis a pivotal pathway for regulating metastasis PMID 33262521
Soluble Guanylate Cyclase Stimulator Vericiguat Attenuates Angiotensin II
Daimuron 42609
Desulfovibrio desulfuricans and its derived metabolites confer resistance to FOLFOX through METTL3 PMID 38484555
外胚层神经皮层 1（ENC1）基因
Platycodin D Ameliorates Cognitive Impairment in Type 2 Diabetes Mellitus Mice via Regulating PI3K/Akt/GSK3β Signaling Pathway PMID 38491972
Apolipoprotein E COG 133 mimetic peptide improves 5
NTRK2 activation cooperates with PTEN deficiency in T
Technical Support
Overcoming PEG─Protein Mutual Repulsion to Improve the Efficiency of PEGylation PMID 36306195
4
Effect of a platelet
Thalidomide
3’,5’
Valyllysine 22677
In vitro activity of retapamulin against linezolid and methicillin
P 450s u nder Re striction (PURE) Screen Using HepaRG and Primary Human Hepatocytes for Discovery of Novel HBV Antivirals PMID 33062174
Cholangiocarcinoma PDHA1 succinylation suppresses macrophage antigen presentation via alpha
Analeptic effects of centrally injected TRH and analogues of TRH in the pentobarbitone
Rapid and reversible relocalization of heat shock factor 1 within seconds to nuclear stress granules PMID 10359787
α
The mechanism of YAP/TAZ transactivation and dual targeting for cancer therapy PMID 40274828
Azido
Desthiobiotin polyethyleneoxide iodoacetamide
NECAP1 Human Pre
Different muscarinic receptor subtypes mediating the phasic activity and basal tone of pig isolated intravesical ureter PMID 7905771
Neuraminidase Inhibitors from the Roots of Caragana sinica PMID 32996697
High
Unveiling the signal valve specifically tuning the TGF
Behavioral and neurophysiological effects of Ro 10
蛋白磷酸酶 3 调节亚基 B，α（PPP3R1）基因
Involvement of Acylated Homoserine Lactones (AHLs) of Aeromonas sobria in Spoilage of Refrigerated Turbot (Scophthalmus maximus L.) PMID 27420072
高尔基磷蛋白 3 样（GOLPH3L）基因
Discovery of a First
Xantphos 161265
A 16 amino acid synthetic peptide derived from human C3d triggers proliferation and specific tyrosine phosphorylation of transformed CR2
T3
Mitoquinone does not improve sperm cryo
Animal
MC
Metabolites of antibody
L
DNA protein cross
Synthesis and biological evaluation of 3
Chlorobutanol maternal serum levels and placental transfer in the mouse PMID 9311085
Hepatitis C virus entry PMID 23463198
Human beta
Krt8 Rat Pre
Polymorphs, co
Effect of Pantethine on Ovarian Tumor Progression and Choline Metabolism PMID 27900284
Antitumor activity of a 5T4 targeting antibody drug conjugate with a novel payload derived from MMAF via C
New Selective Inhibitors of ERG Positive Prostate Cancer ERGi
New haliangicin isomers, potent antifungal metabolites produced by a marine myxobacterium PMID 14513906
Tumor necrosis factor α
Metabolic products of microorganisms. 185. The anthraquinones of the Aspergillus glaucus group. I. Occurrence, isolation, identification and antimicrobial activity PMID 7406630
Positron emission tomography measurement of brain MAO
Cd276 Rat Pre
Palazestrant 2092925
The tricyclic antidepressant clomipramine increases plasma glucose levels of mice PMID 14501155
A method for screening for various sedative
(S)
Implant
EIDD
On
PD
SB 242084 dihydrochloride 1049747
Fas 配体（FASLG）基因
Chemical modulation of chaperone
Antibiofilm agent
SQ
The modulation of fragile X behaviors by the muscarinic M4 antagonist, tropicamide PMID 21942438
Production of a novel neuropeptide encoded by the calcitonin gene via tissue
Cucurbitacin E inhibits cellular proliferation and induces apoptosis in melanoma by suppressing HSDL2 expression PMID 35193614
A new amide from Asarum forbesii Maxim PMID 15621594
Down
Flavonoid constituents from Glycyrrhiza glabra hairy root cultures PMID 11140606
5
Gadobutrol PMID 20641787
DING proteins from phylogenetically different species share high degrees of sequence and structure homology and block transcription of HIV
Chemical perturbation of Mcl
GR231118 (1229U91) and other analogues of the C
Discovery of DS79932728 A Potent, Orally Available G9a/GLP Inhibitor for Treating β
Semisynthesis of natural flavones inhibiting tubulin polymerization, from hesperidin PMID 20356063
Norepinephrine transporter regulation mediates the long
A thioredoxin reductase 1 inhibitor pyrano [3,2
A noncompetitive BACE1 inhibitor TAK
Decarestrictin A1 127393
CP
吲哚胺 2 ,3
Metabolism and disposition of alpha
1
Evaporative light scattering detection of pyrrolizidine alkaloids PMID 14979525
Discovery of a Novel Series of N
Heteroclitin G 144027
XBP1 modulates endoplasmic reticulum and mitochondria crosstalk via regulating NLRP3 in renal ischemia/reperfusion injury PMID 36801911
Raffinose increases autophagy and reduces cell death in UVB
Interference by bovine serum albumin in PED6 based phospholipase A2 screening assays PMID 23210248
BW 723C86, a 5
WAY
BTN2A1 蛋白, Human (Biotinylated, HEK293, Fc
Discovery of a novel water
VH
4
MD2
Tetrahydrocarboline analogs as MCH
ITGB6 蛋白, Human (HEK293, His)
Down regulation of serotonin
Penicillin causes non
Sin3b Rat Pre
PD 116,948, a highly selective A1 adenosine receptor antagonist PMID 3807648
NFATC3 Human Pre
Butamirate 18109
Evaluation of α
ABCE1 的 YAE1 成熟因子（YAE1）基因
Tigogenin inhibits adipocytic differentiation and induces osteoblastic differentiation in mouse bone marrow stromal cells PMID 17363141
Androsterone
BL
Development and application of a rapid and sensitive liquid chromatography
The Role of Sphingomyelin Metabolism in the Protection of Rat Brain Microvascular Endothelial Cells by Mild Hypothermia PMID 34508278
Cynaroside prevents macrophage polarization into pro
V023
Dehydrocorydaline Protects Against Sepsis
Cortical spreading depolarisation
Translation Termination Factor GSPT1 Is a Phenotypically Relevant Off
Galectin
Design and synthesis of novel JNK inhibitors targeting liver pyruvate kinase for the treatment of non
JPHM
Il1rap
Activity of the novel BCR kinase inhibitor IQS019 in preclinical models of B
PKHB1, a thrombospondin
Aticaprant (Standard) (CERC
Role of TGF
ICAM3 抗体 (YA3009)（ICAM3 Antibody (YA3009)）
Exposure to Di
碳水化合物磺基转移酶 5（CHST5）基因
Peptides that mimic the pseudosubstrate region of protein kinase C bind to acidic lipids in membranes PMID 1883933
MCE
Wilforol C 168254
Pomalidomide 4'
Mesenchymal stem cells overexpressing neuropeptide S promote the recovery of rats with spinal cord injury by activating the PI3K/AKT/GSK3β signaling pathway PMID 40022159
MAO
Novel Pro
KRT15 Human Pre
RORγt inverse agonist TF
CHIR 4531 158198
Vinburnine Sensitizes Radiotherapy Efficacy in Nasopharyngeal Carcinoma by Triggering Pyroptosis and Immune Responses via Activation of EDAR
DCG
NAE
Reproductive and developmental toxicity of the herbicide Betanal® Expert and corresponding active ingredients to Daphnia spp PMID 27023815
Leriglitazone
T 盒转录因子 2（TBX2）基因
Estrone 3
MI
Combinatorial development of nebulized mRNA delivery formulations for the lungs PMID 37985700
Phase II trial of AKT inhibitor MK
Remodeling of the Fission Yeast Cdc42 Cell
Activation of Disulfide Redox Switch in REDD1 Promotes Oxidative Stress Under Hyperglycemic Conditions PMID 36170669
Effects of aldicarb and propoxur on cytotoxicity and lipid peroxidation in CHO
Structure
Deguelin, an Akt inhibitor, down
Pharmacokinetic study of pyridinol carbamate in chronic renal insufficiency PMID 6745304
Age
同源框 C5（HOXC5）基因
Bromoxynil 1689
Real time analysis of the affinity regulation of alpha 4
Role of 5
Geranylgeranyltransferase I inhibitor GGTI
Discovery of 12 (BMS
Synthesis of 15
S32826, a nanomolar inhibitor of autotaxin discovery, synthesis and applications as a pharmacological tool PMID 18755937
Analysis of doramectin in the serum of repeatedly treated pastured cattle used to predict the probability of cattle fever ticks (Acari Ixodidae) feeding to repletion PMID 22349982
Hypocretin
A Mucin 16 bispecific T cell
Triterpenoid saponins from Bellis bernardii PMID 8904843
Small molecule RITA binds to p53, blocks p53
Biological activities and safety data of kojic acid and its derivatives A review PMID 35960194
VEGFR
Novel substituted 9
The role of TGF
Ribosome biogenesis in cancer new players and therapeutic avenues PMID 29192214
Identification of Small Molecules that Selectively Inhibit Fluconazole
Structural polysaccharide PCP1 from Polygonatum cyrtonema Hua attenuates atherosclerosis via dual
Anti
I
The combined activation of KCa3.1 and inhibition of Kv11.1/hERG1 currents contribute to overcome Cisplatin resistance in colorectal cancer cells PMID 29161243
Liver governs adipose remodelling via extracellular vesicles in response to lipid overload PMID 32024826
Supplemental carvacrol can reduce the severity of inflammation by influencing the production of mediators of inflammation PMID 25416233
Anticancer activity of the thiosemicarbazones that are based on di
Aristolactam BIII 53948
Tyrosine Kinase 2
Biochemical investigations of the mechanism of action of small molecules ZL006 and IC87201 as potential inhibitors of the nNOS
Anti
IP2 2247640
Pranlukast
Discovery of phenylpyrrolidine derivatives as a novel class of retinol binding protein 4 (RBP4) reducers PMID 34953340
Fibrinogen drives neuroinflammation and neuropathology in perioperative neurocognitive disorders PMID 41273843
Toxicology of indecainide hydrochloride after intravenous administration to rats and dogs PMID 4035704
DPPC
Arrb2 promotes endothelial progenitor cell
Activation of multiple apoptotic pathways in human nasopharyngeal carcinoma cells by the prenylated isoflavone, osajin PMID 21532751
Characterization and mutation analysis of human LEFTY A and LEFTY B, homologues of murine genes implicated in left
Discovery of a Highly Potent and Selective Inhibitor Targeting Protein Lysine Methyltransferase NSD2 PMID 39230932
肌钙蛋白 T1，慢骨骼型（TNNT1）基因
Oroxylin A inhibits glycolysis
Antimicrobial peptides for bone tissue engineering Diversity, effects and applications PMID 36277377
Isolation and Identification of Saponins from the Natural Pasturage Asterothamnus centrali
Imeglimin 775351
pGlu
(2S,3R)
A Combination of Cardamonin and Doxorubicin Selectively Affect Cell Viability of Melanoma Cells An In Vitro Study PMID 39061932
The selective 5
Light
The 67
Stereo
Discovery and evaluation of ZT55, a novel highly
Enantioselective Synthesis of (
The selective lipoprotein
Synthesis, Anticancer Evaluation, and Molecular Docking of Triazolylmethyl
A nanomolar
Kinetic analysis of the interaction of tissue transglutaminase with a nonpeptidic slow
Interleukin
(S)
Biliary excretion and pharmacokinetics of a gadolinium chelate used as a liver
WCF
Complement Cross Talks With H
AChE
Novel glycosyl prodrug of RXP03 as MMP
DDX24 Mutation Alters NPM1 Phase Behavior and Disrupts Nucleolar Homeostasis in Vascular Malformations PMID 37705750
Discovery of novel non
N
OMTX705, a Novel FAP
Zea mays
KBH
Effects of various penetration enhancers on penetration of aminophylline through shed snake skin PMID 24644435
apoptotic responses
VAL
Overexpression of MCL1 attenuates irritable bowel syndrome by regulating cuproptosis Screening and validation PMID 39488085
Discovery of a Potent and Selective ATAD2 Bromodomain Inhibitor with Antiproliferative Activity in Breast Cancer Models PMID 35133824
Antimicrobial activity of extracts and some compounds from Calea platylepis PMID 15261392
Structure determination of new analogues of vardenafil and sildenafil in dietary supplements PMID 17364912
Suppression of c
TERT's protective effect on trophoblast cells Reducing mitochondrial ROS PMID 40139512
hsa
纤连蛋白 III 型和锚蛋白重复结构域 1（FANK1）基因
PSFL 2915
Antitumor activity of S116836, a novel tyrosine kinase inhibitor, against imatinib
Discovery of benzimidazole
microRNA
UAB116
Activation of Sirt1 protects from single
Optimization of New Catalytic Topoisomerase II Inhibitors as an Anti
The inflammatory cytokines TWEAK and TNFα reduce renal klotho expression through NFκB PMID 21719790
Induced optical activity of various aminoacridines bound to DNA PMID 6063543
NecroX
N
Identification of Ribosomal Protein S4, Y
Cross
(Tyr1)
肌球蛋白集成电路（MYO1C）基因
Cardioprotective effect of SMND
Inhibition of a Golgi complex lysophospholipid acyltransferase induces membrane tubule formation and retrograde trafficking PMID 12925777
Escin alleviates peripheral neuropathy in streptozotocin induced diabetes in rats PMID 32407839
EGFR
PL
MCE
SNAP 398299 903878
(E,E)
Reduced chemokine C
EPH 受体 B3（EPHB3）基因
IGF2 modulates the microenvironment for osteoclastogenesis PMID 19056348
Mesaconitine 2752
2'
terminal alkyne
SM51a 2764770
PCSK9
siRNA drug delivery across the blood
Mechanism of inhibition for N6022, a first
Spirostan
Phenotypic Differences in Primary Murine Microglia Treated with NOD1, NOD2, and NOD1/2 Agonists PMID 31907866
(S)
YL 5092
Design, Synthesis, and Herbicidal Activity of Substituted 3
Intervention of exogenous VEGF protect brain microvascular endothelial cells from hypoxia
Sebuthylazine 7286
Design, synthesis, and biological evaluation of chalcone acetamide derivatives against triple negative breast cancer PMID 38750906
DM1
E913 342394
Effect of E5324, a novel inhibitor of acyl
Discovery of Clinical Candidate 2
Daphmacropodine 39729
Verapamil
Echinacoside suppresses macrophage lipid accumulation and attenuates atherosclerosis via the MDM2/PPARγ/ABCA1 signaling axis PMID 40819820
Cisplatin Protein Binding Partners and Their Relevance for Platinum Drug Sensitivity PMID 32466394
m
Lonidamine, a Novel Modulator for the BvgAS System of Bordetella Species PMID 39674913
Exploring the Mechanism of Ferroptosis Induction by Sappanone A in Cancer Insights into the Mitochondrial Dysfunction Mediated by NRF2/xCT/GPX4 Axis PMID 39430236
α
GSK364735
Selective Inhibition of MMP
Sporminarin A 915403
Stronger Uricosuric Effects of the Novel Selective URAT1 Inhibitor UR
beta
Expression and characterization of jingzhaotoxin
BMS
Methyltriphenylphosphonium iodide
Tri
Knockdown of Oligosaccharyltransferase Subunit Ribophorin 1 Induces Endoplasmic
Indicine
Exploration of allosteric agonism structure
1,10
Preclinical efficacy of the novel competitive NAMPT inhibitor STF
The Glutamate Dehydrogenase Pathway and Its Roles in Cell and Tissue Biology in Health and Disease PMID 28208702
W4275 3051650
TRPM7 Upregulate the Activity of SMAD1 through PLC Signaling Way to Promote Osteogenesis of hBMSCs PMID 32596398
Hit Selection of Dipeptidyl Peptidase
Selectivity of LG50643 for postjunctional muscarinic
The cannabinoid antagonist SR144528 enhances the acute effect of WIN 55,212
CD2 augmentation enhances CAR
LY56110 26766
SKA
Imeglimin prevents human endothelial cell death by inhibiting mitochondrial permeability transition without inhibiting mitochondrial respiration PMID 27551496
Responses of AChE and GST activities to insecticide coexposure in Carassius auratus PMID 20549641
Purine phosphoribosyltransferase
Chimonanthine 5545
Mip
Naturally occurring monoepoxides of eicosapentaenoic acid and docosahexaenoic acid are bioactive antihyperalgesic lipids PMID 20664072
An Essential Role for the Tetraspanin LHFPL4 in the Cell
AFM32a hydrochloride 2988594
Des
Oroxylin A inhibits colitis
24 Bisphenol S
DGAT
Metabolic profiles for the pyrrolizidine alkaloid neopetasitenine and its metabolite petasitenine in humans extrapolated from rat in vivo and in vitro data sets using a simplified physiologically based pharmacokinetic model PMID 34470991
Plasma membrane monoamine transporters structure, regulation and function PMID 12511858
Copovidone (50% in ethanol) 25086
Dopamine D3 receptor ligand
ME 3407 133903
Arenobufagin, a natural bufadienolide from toad venom, induces apoptosis and autophagy in human hepatocellular carcinoma cells through inhibition of PI3K/Akt/mTOR pathway PMID 23393227
UBP684 1357838
β2AR ligand 1 3051498
Olitigaltin 1450824
Fragment
4
Hemsloside H1 102146
Bst1/CD157
D
Halogenated diarylacetylenes repress c
Kojic acid applications in cosmetic and pharmaceutical preparations PMID 30537675
Phase II, randomized, double
Lack of genotoxic effect of food dyes amaranth, sunset yellow and tartrazine and their metabolites in the gut micronucleus assay in mice PMID 19095036
Primula spectabilis Tratt. aerial parts morphology, volatile compounds and flavonoids PMID 21612805
Engineered Aminoacyl
Astrapterocarpan isolated from Astragalus membranaceus inhibits proliferation of vascular smooth muscle cells PMID 16297381
Rational design, synthesis and testing of novel tricyclic topoisomerase inhibitors for the treatment of bacterial infections part 2 PMID 34095845
Determination of rabeprazole and its active metabolite, rabeprazole thioether in human plasma by column
New pyridazinone
Synthesis and antiviral activity of cyclopropyl
Aldehyde
Discovery of novel 5
Combined toxicity of trifloxystrobin and fluopyram to zebrafish embryos and the effect on bone development PMID 38281391
Fosinoprilat alleviates lipopolysaccharide (LPS)
Carvacrol Induced Program Cell Death and Cell Cycle Arrest in Androgen
A pan
Esterastin, an inhibitor of esterase, produced by actinomycetes PMID 567214
Ubiquitin specific peptidase 19 is a prognostic biomarker and affect the proliferation and migration of clear cell renal cell carcinoma PMID 32236633
Eresepine
Sappanone A inhibits RANKL
Synthesis and biological evaluation of 4
Diversity of locally produced IFN
2,6
(R)
From the selective serotonin transporter inhibitor citalopram to the selective norepinephrine transporter inhibitor talopram synthesis and structure
Amino Acid Metabolism
ALS2
Gpc1
Isoflupredone
MCE
Plasminogen activator inhibitor
(R)
6764
Ang
A truncated HIV
Discovery of 1,2,3,4
Antibacterial activity and pharmacokinetic profile of a promising antibacterial agent 14
Development of Novel Small Antitumor Compounds Inhibiting PD
Eupatobenzofuran 1275622
Stem cell membrane
Hemorphin 7 reflects hemoglobin proteolysis in abdominal aortic aneurysm PMID 19910633
[D
T 细胞急性淋巴细胞白血病
Mitoquinone mesylate promotes oocyte maturation and subsequent embryonic development by regulating oxidative stress in Tibetan sheep PMID 40424944
Benzyloxy carbonyl
Inhibition of aryl hydrocarbon receptor signaling promotes the terminal differentiation of human erythroblasts PMID 35022784
Mesembrenone
Remdesivir intermediate
NPN
Enhanced Cuproptosis via Metabolic Reprogramming Using Copper
CD127/IL
MK
Tetrahydroberberine, an isoquinoline alkaloid isolated from corydalis tuber, enhances gastrointestinal motor function PMID 21659472
N
Y36912
MK 0429
Pox viral vaccine approaches PMID 16338420
SARS
TP
Thalidomide
Endothelin
Δ4
Diallyl sulfide protects against lipopolysaccharide/d
acceptor
核糖体蛋白 S5（RPS5）基因
New potent and selective polyfluoroalkyl ketone inhibitors of GVIA calcium
Metronidazole
Comparative evaluation of central muscarinic receptor binding activity by oxybutynin, tolterodine and darifenacin used to treat overactive bladder PMID 17222678
Ginsenoside mRb
Vitamin B12 protects against superoxide
Pank1 Rat Pre
HDAC
Reviving the guardian of the genome Small molecule activators of p53 PMID 28351719
Zuclomiphene 15690
BRD9526
Antimicrobial activity of prulifloxacin in comparison with other fluoroquinolones against community
Potent and long
Development of AC265347
Fostamatinib Disodium 1025687
Propan
Discovery of antileishmanial hits in the 3
Piboserod hydrochloride 178273
Finding the Right Heavy Chains for Immunostimulatory Antibodies PMID 36142278
Cancer chemotherapy by liposomal 6
(D
Benzo(a)pyrene induced lung cancer Role of dietary phytochemicals in chemoprevention PMID 26398396
New hepatoprotective isoflavone glucosides from Pueraria lobata (Willd.) Ohwi PMID 29968479
Design, synthesis, and biological evaluation of potent 1,2,3,4
Illudin S 1149
1H
1,4
GPR40 partial agonists and AgoPAMs Differentiating effects on glucose and hormonal secretions in the rodent PMID 29053717
Discovery of Orally Bioavailable Phthalazinone Analogues as an ENPP1 Inhibitor for STING
Metabolism of propranolol during percutaneous absorption in human skin PMID 8377110
Old drug, new indication Olsalazine sodium reduced serum uric acid levels in mice via inhibiting xanthine oxidoreductase activity PMID 29132796
Design, synthesis, and pharmacological evaluation of novel and selective COX
HET
CD1B
XC 基序趋化因子配体 2（XCL2）基因
α
(S,S)
Bpi
4
Novel benzothiazole/benzothiazole thiazolidine
Interleukin
PRMT5
DOCK2 抗体 (YA8613)（DOCK2 Antibody (YA8613)）
The Small Non
Opioid activities of human beta
AWD 12
4
Lanatoside C protects mice against bleomycin
MCE
ML251 1486482
Highly Potent Immunotoxins Targeting the Membrane
Regulation of molecular chaperone gene transcription involves the serine phosphorylation, 14
PF
Deguelin exerts anticancer activity of human gastric cancer MGC
Identification of IMP Dehydrogenase as a Potential Target for Anti
Mitochondrial Dysfunctions Regulated Radioresistance through Mitochondria
SARS
The biosynthesis of isopimpinellin PMID 890566
Escin suppresses immune cell infiltration and selectively modulates Nrf2/HO
Interactions between PHD3
MCE
Comparative in vitro activity profiles of novel bis
Angiotensin II type 1 receptor (181
Phosphatase
Azido sphingosine (d14 1)
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